[1,2,4]triazolo[4,3-a]phthalazines: inhibitors of diverse bromodomains.

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Published in J Med Chem on December 30, 2013

Authors

Oleg Fedorov1, Hannah Lingard, Chris Wells, Octovia P Monteiro, Sarah Picaud, Tracy Keates, Clarence Yapp, Martin Philpott, Sarah J Martin, Ildiko Felletar, Brian D Marsden, Panagis Filippakopoulos, Susanne Müller, Stefan Knapp, Paul E Brennan

Author Affiliations

1: Structural Genomics Consortium, Nuffield Department of Medicine, University of Oxford , Old Road Campus Research Building, Roosevelt Drive, Oxford OX3 7DQ, U.K.

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