The structure-activity relationships of L3MBTL3 inhibitors: flexibility of the dimer interface.

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Published in Medchemcomm on November 01, 2013

Authors

Michelle A Camerino1, Nan Zhong2, Aiping Dong2, Bradley M Dickson1, Lindsey I James1, Brandi M Baughman1, Jacqueline L Norris1, Dmitri B Kireev1, William P Janzen1, Cheryl H Arrowsmith3, Stephen V Frye1

Author Affiliations

1: Center for Integrative Chemical Biology and Drug Discovery, Division of Chemical Biology and Medicinal Chemistry, University of North Carolina Eshelman School of Pharmacy University of North Carolina at Chapel Hill, Chapel Hill, North Carolina, USA. ; Tel: (919) 843-5486.
2: Structural Genomics Consortium, University of Toronto, Ontario, Canada.
3: Center for Integrative Chemical Biology and Drug Discovery, Division of Chemical Biology and Medicinal Chemistry, University of North Carolina Eshelman School of Pharmacy University of North Carolina at Chapel Hill, Chapel Hill, North Carolina, USA. ; Tel: (919) 843-5486 ; Structural Genomics Consortium, University of Toronto, Ontario, Canada ; Department of Medical Biophysics, University of Toronto Ontario, Canada ; Princess Margaret Cancer Centre, 101 College Street, Toronto, Ontario, Canada, M5G 1L7.

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