The TLQP-21 peptide activates the G-protein-coupled receptor C3aR1 via a folding-upon-binding mechanism.

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Published in Structure on November 13, 2014

Authors

Cheryl Cero1, Vitaly V Vostrikov2, Raffaello Verardi2, Cinzia Severini3, Tata Gopinath2, Patrick D Braun4, Maria F Sassano5, Allison Gurney1, Bryan L Roth5, Lucy Vulchanova6, Roberta Possenti3,7, Gianluigi Veglia2, Alessandro Bartolomucci1

Author Affiliations

1: Department of Integrative Biology and Physiology, University of Minnesota, Minneapolis, MN 55455.
2: Department of Biochemistry, Molecular Biology and Biophysics, University of Minnesota, Minneapolis, MN 55455.
3: Institute of Cell Biology and Neurobiology, National Research Council, Rome, Italy 00143.
4: Department of Pharmaceutics, University of Minnesota, Minneapolis, MN 55455.
5: Department of Pharmacology and National Institute of Mental Health Psychoactive Drug Screening Program School of Medicine, University of North Carolina, Chapel Hill, NC 27599.
6: Department of Veterinary and Biomedical Sciences, University of Minnesota, Saint Paul, MN 55108.
7: Department of Medicine of System, University of Rome 'Tor Vergata', Rome, Italy 00133.

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