Characterization of RA839, a Noncovalent Small Molecule Binder to Keap1 and Selective Activator of Nrf2 Signaling.

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Published in J Biol Chem on October 12, 2015

Authors

Angelika F Winkel1, Christian K Engel1, Daniel Margerie1, Aimo Kannt2, Hauke Szillat1, Heiner Glombik1, Christopher Kallus1, Sven Ruf1, Stefan Güssregen1, Jens Riedel1, Andreas W Herling1, Andreas von Knethen3, Andreas Weigert3, Bernhard Brüne3, Dieter Schmoll4

Author Affiliations

1: From the R&D, Sanofi, 65926 Frankfurt, Germany.
2: From the R&D, Sanofi, 65926 Frankfurt, Germany, the Medical Faculty Mannheim, Heidelberg University, 69120 Mannheim, Germany.
3: the Faculty of Medicine, Biochemistry I, Goethe-University Frankfurt, 60590 Frankfurt, Germany.
4: From the R&D, Sanofi, 65926 Frankfurt, Germany, dieter.schmoll@sanofi.com.

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