Optimization of the Solubility of HIV-1-Neutralizing Antibody 10E8 through Somatic Variation and Structure-Based Design.

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Published in J Virol on June 10, 2016

Authors

Young D Kwon1, Ivelin S Georgiev1, Gilad Ofek1, Baoshan Zhang1, Mangaiarkarasi Asokan1, Robert T Bailer1, Amy Bao1, William Caruso1, Xuejun Chen1, Misook Choe1, Aliaksandr Druz1, Sung-Youl Ko1, Mark K Louder1, Krisha McKee1, Sijy O'Dell1, Amarendra Pegu1, Rebecca S Rudicell1, Wei Shi1, Keyun Wang1, Yongping Yang1, Mandy Alger1, Michael F Bender1, Kevin Carlton1, Jonathan W Cooper1, Julie Blinn2, Joshua Eudailey2, Krissey Lloyd2, Robert Parks2, S Munir Alam2, Barton F Haynes2, Neal N Padte3, Jian Yu3, David D Ho3, Jinghe Huang4, Mark Connors4, Richard M Schwartz1, John R Mascola5, Peter D Kwong5

Author Affiliations

1: Vaccine Research Center, National Institute of Allergy and Infectious Diseases, National Institutes of Health, Bethesda, Maryland, USA.
2: Duke Human Vaccine Institute, Departments of Medicine, Surgery, Pediatrics and Immunology, Duke University School of Medicine, Durham, North Carolina, USA Center for HIV/AIDS Vaccine Immunology-Immunogen Discovery, Duke University, Durham, North Carolina, USA.
3: The Aaron Diamond AIDS Research Center, Rockefeller University, New York, New York, USA.
4: HIV-Specific Immunity Section, Laboratory of Immunoregulation, National Institute of Allergy and Infectious Diseases, National Institutes of Health, Bethesda, Maryland, USA.
5: Vaccine Research Center, National Institute of Allergy and Infectious Diseases, National Institutes of Health, Bethesda, Maryland, USA jmascola@mail.nih.gov pdkwong@nih.gov.

Associated clinical trials:

VRC 610: Phase I Safety and Pharmacokinetics Study to Evaluate a Human Monoclonal Antibody (MAB) VRC-HIVMAB095-00-AB (10E8VLS) Administered Alone or Concurrently With MAB VRC- HIVMAB075-00-AB (VRC07-523LS) Via Subcutaneous Injection in Healthy Adults | NCT03565315

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