Regulation of HIF1α under Hypoxia by APE1/Ref-1 Impacts CA9 Expression: Dual Targeting in Patient-Derived 3D Pancreatic Cancer Models.

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Published in Mol Cancer Ther on August 17, 2016

Authors

Derek P Logsdon1, Michelle Grimard2, Meihua Luo2, Safi Shahda3,4, Yanlin Jiang2, Yan Tong5, Zhangsheng Yu5, Nicholas Zyromski4,6, Ernestina Schipani7, Fabrizio Carta8, Claudiu T Supuran8, Murray Korc4,9,10, Mircea Ivan3,4,11, Mark R Kelley1,2,4,10, Melissa L Fishel12,2,4

Author Affiliations

1: Department of Pharmacology and Toxicology, Indiana University School of Medicine, Indianapolis, Indiana.
2: Department of Pediatrics, Wells Center for Pediatric Research, Indiana University School of Medicine, Indianapolis, Indiana.
3: Division of Hematology/Oncology, Department of Medicine, Indiana University School of Medicine, Indianapolis, Indiana.
4: Pancreatic Cancer Signature Center, Indianapolis, Indiana.
5: Department of Biostatistics, Indiana University School of Medicine, Indianapolis, Indiana.
6: Department of Surgery, Indiana University School of Medicine, Indianapolis, Indiana.
7: Department of Orthopaedic Surgery, University of Michigan, Ann Arbor, Michigan.
8: Neurofarba Department, Section of Medicinal Chemistry, University of Florence, Florence, Italy.
9: Division of Endocrinology, Department of Medicine, Indiana University School of Medicine, Indianapolis, Indiana.
10: Department of Biochemistry and Molecular Biology, Indiana University School of Medicine, Indianapolis, Indiana.
11: Department of Microbiology and Immunology, Indiana University School of Medicine, Indianapolis, Indiana.
12: Department of Pharmacology and Toxicology, Indiana University School of Medicine, Indianapolis, Indiana. mfishel@iu.edu.

Associated clinical trials:

Safety Study of SLC-0111 in Subjects With Advanced Solid Tumours | NCT02215850

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