Stereospecific Palladium-Catalyzed C-H Arylation of Pyroglutamic Acid Derivatives at the C3 Position Enabled by 8-Aminoquinoline as a Directing Group.

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🔗 View Article (PMID 28809506)

Published in Org Lett on August 15, 2017

Authors

Oscar Verho¹^,2, Micah Maetani¹^,2, Bruno Melillo¹^,2, Jochen Zoller¹^,2, Stuart L Schreiber³

Author Affiliations

1: Department of Chemistry and Chemical Biology, Harvard University , Cambridge, Massachusetts 02138, United States.
2: Broad Institute , Cambridge, Massachusetts 02142, United States.
3: Department of Chemistry and Chemical Biology, Howard Hughes Medical Institute, Harvard University, Cambridge, United States.

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