Published in Am J Physiol on June 01, 1985
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Covalent binding of a selective agonist irreversibly activates guinea pig coronary artery A2 adenosine receptors. Naunyn Schmiedebergs Arch Pharmacol (1993) 0.94
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Protection against infarction afforded by preconditioning is mediated by A1 adenosine receptors in rabbit heart. Circulation (1991) 4.30
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8-Cyclopentyl-1,3-dipropylxanthine (DPCPX)--a selective high affinity antagonist radioligand for A1 adenosine receptors. Naunyn Schmiedebergs Arch Pharmacol (1987) 1.99
Evidence that the adenosine A3 receptor may mediate the protection afforded by preconditioning in the isolated rabbit heart. Cardiovasc Res (1994) 1.62
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Structure-activity relationships for N6-substituted adenosines at a brain A1-adenosine receptor with a comparison to an A2-adenosine receptor regulating coronary blood flow. Biochem Pharmacol (1986) 1.39
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Changes in content of purine nucleoside in canine myocardium during coronary occlusion. Circ Res (1970) 1.28
Evidence for an adenosine receptor on the surface of dog coronary myocytes. Circ Res (1976) 1.24
A simple, specific, radioisotopic assay for 5'-nucleotidase. Anal Biochem (1975) 1.24
Characterization of the A1 adenosine receptor-adenylate cyclase system of cerebral cortex using an agonist photoaffinity ligand. J Neurochem (1986) 1.21
Definition of subclasses of adenosine receptors associated with adenylate cyclase: interaction of adenosine analogs with inhibitory A1 receptors and stimulatory A2 receptors. Can J Physiol Pharmacol (1987) 1.16
Endothelial cell uptake of adenosine in canine skeletal muscle. Am J Physiol (1986) 1.16
Dog coronary artery adenosine receptor: structure of the N6-alkyl subregion. J Med Chem (1985) 1.11
Characterization of two affinity states of adenosine A2a receptors with a new radioligand, 2-[2-(4-amino-3-[125I]iodophenyl)ethylamino]adenosine. Mol Pharmacol (1995) 1.06
N6-substituted N-alkyladenosine-5'-uronamides: bifunctional ligands having recognition groups for A1 and A2 adenosine receptors. J Med Chem (1986) 1.06
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2-Alkoxyadenosines: potent and selective agonists at the coronary artery A2 adenosine receptor. J Med Chem (1991) 1.02
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Coronary vasoactivity of adenosine in the conscious dog. Circ Res (1979) 1.00
Metabolic control of coronary blood flow. Prog Cardiovasc Dis (1987) 0.98
Intracoronary adenosine deaminase reduces canine myocardial reactive hyperemia. Circ Res (1981) 0.98
Covalent binding of a selective agonist irreversibly activates guinea pig coronary artery A2 adenosine receptors. Naunyn Schmiedebergs Arch Pharmacol (1993) 0.94
Effect of aminophylline on adenosine and exercise dilation of rat cremaster arterioles. Am J Physiol (1984) 0.94
Myocardial reactive hyperemia. Circ Res (1975) 0.93
Activity of N6-substituted 2-chloroadenosines at A1 and A2 adenosine receptors. J Med Chem (1991) 0.92
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N6,9-disubstituted adenines: potent, selective antagonists at the A1 adenosine receptor. J Med Chem (1991) 0.91
Inhibition of platelet aggregation by adenosine receptor agonists. Naunyn Schmiedebergs Arch Pharmacol (1994) 0.91
Adenosine metabolism in canine myocardial reactive hyperemia. Circ Res (1978) 0.91
Structure-activity relationships for 2-substituted adenosines at A1 and A2 adenosine receptors. Pharmacology (1993) 0.90
Adenosine uptake by canine heart. Circ Res (1972) 0.90
2-Phenylethoxy-9-methyladenine: an adenosine receptor antagonist that discriminates between A2 adenosine receptors in the aorta and the coronary vessels from the guinea pig. J Pharmacol Exp Ther (1993) 0.90
Functional characterization of adenosine A2 receptors in Jurkat cells and PC12 cells using adenosine receptor agonists. Naunyn Schmiedebergs Arch Pharmacol (1996) 0.89
Dog coronary artery adenosine receptor: structure of the N6-aryl subregion. J Med Chem (1986) 0.89
Adenosine analogs mediating depressant effects on synaptic transmission in rat hippocampus: structure-activity relationships for the N6 subregion. Naunyn Schmiedebergs Arch Pharmacol (1986) 0.89
Age-associated alterations in myocardial contractile properties. Am J Physiol (1972) 0.88
Substituted 1,3-dipropylxanthines as irreversible antagonists of A1 adenosine receptors. J Med Chem (1994) 0.87
Nitric oxide modulates coronary autoregulation in the guinea pig. Circ Res (1992) 0.87
Dose-dependent increase in sensitivity to calcium-induced mitochondrial dysfunction and cardiomyocyte cell injury by doxorubicin. J Mol Cell Cardiol (1996) 0.86
Transcapillary adenosine transport in isolated guinea pig and rat hearts. Am J Physiol (1990) 0.86
Normal absorption in Thai subjects with non-specific jejunal abnormalities. Br Med J (1967) 0.86
2-(N'-alkylidenehydrazino)adenosines: potent and selective coronary vasodilators. J Med Chem (1992) 0.86
Cardiovascular actions of adenosines, but not adenosine receptors, differ in rat and guinea pig. Life Sci (1991) 0.84
Local factors regulating cardiac and skeletal muscle blood flow. Annu Rev Physiol (1981) 0.83
Adenosine stimulates phosphate and glucose transport in opossum kidney epithelial cells. Am J Physiol (1991) 0.83
Cyclic adenosine 3',5'-monophosphate-stimulated protein kinase and a substrate associated with cardiac sarcoplasmic reticulum. J Biol Chem (1973) 0.83
Role of adenosine in coronary blood flow regulation after reductions in perfusion pressure. Circ Res (1985) 0.82
The anti-infarct effect of an adenosine A1-selective agonist is diminished after prolonged infusion as is the cardioprotective effect of ischaemic preconditioning in rabbit heart. J Mol Cell Cardiol (1994) 0.82
Adenosine's role in regulating basal coronary arteriolar tone. Am J Physiol (1986) 0.82
N6-substituted 9-methyladenines: a new class of adenosine receptor antagonists. FEBS Lett (1987) 0.82
Mechanical properties of the copper-deficient rat heart. J Nutr (1982) 0.81
2-aralkoxyadenosines: potent and selective agonists at the coronary artery A2 adenosine receptor. J Med Chem (1991) 0.81
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Cardiac muscle mechanics from Doca- and aging spontaneously hypertensive rats. Am J Physiol (1978) 0.80
2-(N'-aralkylidenehydrazino)adenosines: potent and selective coronary vasodilators. J Med Chem (1992) 0.80
A radioligand-binding assay for adenosine in tissue extracts. Anal Biochem (1978) 0.80
Ligand binding to the adenine analogue binding protein of the rabbit erythrocyte. Biochemistry (1978) 0.80
Upregulated renal adenosine A1 receptors augment PKC and glucose transport but inhibit proliferation. Am J Physiol (1996) 0.80
Glibenclamide reduces the coronary vasoactivity of adenosine receptor agonists. J Pharmacol Exp Ther (1994) 0.79
Limitations in predicting oxyhemoglobin saturation of dog blood from PO2. Am J Physiol (1980) 0.79
Relationship of cardiac oxygen usage, adenosine content, and coronary resistance in dogs. Circ Res (1980) 0.79
Metabolic regulation of coronary blood flow. Physiologist (1982) 0.78
Forskolin potentiates the coronary vasoactivity of adenosine in the open-chest dog. Circ Res (1984) 0.78
Compartmentalization of the adenosine pool of dog and rat hearts. Circ Res (1982) 0.78
Coronary vasoactivity of acetate in dog and guinea-pig. Basic Res Cardiol (1986) 0.77
Structure-activity relationship of 2-(ar) alkoxyadenosines at the adenosine A2 receptor in coronary artery. Eur J Pharmacol (1993) 0.77
Role of adenosine in mediating the coronary vasodilative response to acute hypoxia. Cardiovasc Res (1987) 0.77
Selective A2-adenosine receptor agonists do not alter action potential duration, twitch shortening, or cAMP accumulation in guinea pig, rat, or rabbit isolated ventricular myocytes. Circ Res (1993) 0.77
Interference with calcium-dependent mitochondrial bioenergetics in cardiac myocytes isolated from doxorubicin-treated rats. Toxicol Appl Pharmacol (2001) 0.77
Role of adenosine in mediating myocardial blood flow response to isoproterenol: observations in closed chest, sedated, domestic swine. Cardiovasc Res (1986) 0.77
Calcium reintroduction decreases viability of cardiac myocytes from copper-deficient rats. J Nutr (1999) 0.77
Biological activity and a modified synthesis of 8-amino-3-beta-D-ribofuranosyl-1,2,4-triazolo[4,3-a]pyrazine, an isomer of formycin. J Med Chem (1984) 0.76
Mechanical properties of cardiac muscle from spontaneously hypertensive rats: accentuated aftercontractions. Proc Soc Exp Biol Med (1977) 0.76
Adenosine receptor antagonism attenuates angiotensin II effects on adrenergic neurotransmission in the rabbit isolated vas deferens. J Pharmacol Exp Ther (1990) 0.76
Membrane potentials and contractile events of hypertrophied rat cardia muscle. Proc Soc Exp Biol Med (1981) 0.76
Augmented aftercontractions in papillary muscles from rats with cardiac hypertrophy. Am J Physiol (1979) 0.76
Binding of tritiated and radioiodinated ZM241,385 to brain A2A adenosine receptors. Nucl Med Biol (2004) 0.75
Pseudomonas aeruginosa exotoxin A enhances automaticity and potentiates hypoxic depression of isolated rat hearts. Proc Soc Exp Biol Med (1993) 0.75
Effect of adenosine deaminase on myocardial reactive hyperemia: preliminary report. Basic Res Cardiol (1981) 0.75
Myocardial: blood purine nucleoside concentration ratios in canine myocardium. Adv Exp Med Biol (1973) 0.75
Coronary vasoactivity of adenosine covalently linked to polylysine. Life Sci (1977) 0.75
Exercise performance and hemodynamics during dietary potassium depletion in dogs. J Appl Physiol Respir Environ Exerc Physiol (1978) 0.75
Cardiac norepinephrine and intrinsic properties of isolated hypertrophied hearts from DOCA hypertensive rats. J Mol Cell Cardiol (1984) 0.75
Potency of N6 secondary and tertiary alkyladenosine analogues at presynaptic A1 adenosine receptors in guinea-pig ileum. J Auton Pharmacol (1991) 0.75
An implantable semiconductor beta-radiation detector. Am J Physiol (1977) 0.75
Adenosine metabolism: properties of dog heart microsomal 5'-nucleotidase. Adv Exp Med Biol (1973) 0.75
A1 adenosine receptor antagonists as ligands for positron emission tomography (PET) and single-photon emission tomography (SPET). J Med Chem (1998) 0.75
Phenyl(dihydroboryl) polyacrylamide beads for chromatography of ribonucleosides in tissue extracts. J Chromatogr (1979) 0.75
Cardiac hypertrophy in copper-deficient rats is not attenuated by angiotensin II receptor antagonist L-158,809. Proc Soc Exp Biol Med (1996) 0.75
Adenosine regulation of canine cardiac adenylate cyclase. Biochem Pharmacol (1981) 0.75
Cardiac anaphylaxis in isolated guinea pig hearts perfused at constant flow or constant pressure. Proc Soc Exp Biol Med (1987) 0.75
Transient postocclusive renal vasospasm in conscious rhesus monkeys. Am J Physiol (1977) 0.75
Evaluation of radioiodinated 8-Cyclopentyl-3-[(E)-3-iodoprop-2-en-1-yl]-1-propylxanthine ([*I]CPIPX) as a new potential A1 adenosine receptor antagonist for SPECT. Nucl Med Biol (2003) 0.75
Steric requirements for binding of adenosine to a membrane carrier in canine heart. Biochim Biophys Acta (1973) 0.75
Inquiry into hereditary factors in the pathogenesis of dengue haemorrhagic fever: a preliminary note. Bull World Health Organ (1966) 0.75
Factors determining delayed peak flow in canine myocardial reactive hyperaemia. Cardiovasc Res (1979) 0.75
Isovolumetric properties of ventricles of spontaneously hypertensive rats. Am J Physiol (1981) 0.75