Diazoxide and D600 inhibition of insulin release. Distinct mechanisms explain the specificity for different stimuli.

PubWeight™: 1.15‹?› | Rank: Top 10%

🔗 View Article (PMID 6131003)

Published in Diabetes on September 01, 1982

Authors

J C Henquin, S Charles, M Nenquin, F Mathot, T Tamagawa

Articles citing this

Evidence that glucose can control insulin release independently from its action on ATP-sensitive K+ channels in mouse B cells. J Clin Invest (1992) 2.06

Phentolamine and yohimbine inhibit ATP-sensitive K+ channels in mouse pancreatic beta-cells. Br J Pharmacol (1990) 1.45

Mechanisms of ATP release and signalling in the blood vessel wall. Cardiovasc Res (2012) 1.27

Effects of putative activators of K+ channels in mouse pancreatic beta-cells. Br J Pharmacol (1989) 1.17

Block of ATP-regulated potassium channels by phentolamine and other alpha-adrenoceptor antagonists. Br J Pharmacol (1991) 1.16

Stimulation of the KATP channel by ADP and diazoxide requires nucleotide hydrolysis in mouse pancreatic beta-cells. J Physiol (1993) 1.13

The effects of cromakalim on ATP-sensitive potassium channels in insulin-secreting cells. Br J Pharmacol (1990) 1.02

Increase in insulin release from rat pancreatic islets by quinolone antibiotics. Br J Pharmacol (1996) 0.95

Clonidine inhibits ATP-sensitive K+ channels in mouse pancreatic beta-cells. Br J Pharmacol (1991) 0.92

Effects of pinacidil, RP 49356 and nicorandil on ATP-sensitive potassium channels in insulin-secreting cells. Br J Pharmacol (1990) 0.91

Effects of theophylline and dibutyryl cyclic adenosine monophosphate on the membrane potential of mouse pancreatic beta-cells. J Physiol (1984) 0.85

Evidence of a role for GTP in the potentiation of Ca(2+)-induced insulin secretion by glucose in intact rat islets. J Clin Invest (1995) 0.83

Distinct effects of various amino acids on 45Ca2+ fluxes in rat pancreatic islets. Biochem J (1983) 0.82

Cibenzoline inhibits diazoxide- and 2,4-dinitrophenol-activated ATP-sensitive K+ channels in guinea-pig ventricular cells. Br J Pharmacol (1993) 0.78

Different insulin-secretory responses to calcium-channel blockers in islets of lean and obese (ob/ob) mice. Biochem J (1988) 0.75

Articles by these authors

Pancreatic beta-cell mass in European subjects with type 2 diabetes. Diabetes Obes Metab (2008) 3.96

Mechanisms and physiological significance of the cholinergic control of pancreatic beta-cell function. Endocr Rev (2001) 2.92

Cellular composition of the human diabetic pancreas. Diabetologia (1983) 2.71

Significance of ionic fluxes and changes in membrane potential for stimulus-secretion coupling in pancreatic B-cells. Experientia (1984) 2.43

Direct glucocorticoid inhibition of insulin secretion. An in vitro study of dexamethasone effects in mouse islets. J Clin Invest (1997) 2.21

Evidence that glucose can control insulin release independently from its action on ATP-sensitive K+ channels in mouse B cells. J Clin Invest (1992) 2.06

Oscillations of secretion driven by oscillations of cytoplasmic Ca2+ as evidences in single pancreatic islets. J Biol Chem (1993) 1.95

Opposite effects of tolbutamide and diazoxide on 86Rb+ fluxes and membrane potential in pancreatic B cells. Biochem Pharmacol (1982) 1.90

D-glucose inhibits potassium efflux from pancreatic islet cells. Nature (1978) 1.86

An optical spectrum of the afterglow of a gamma-ray burst at a redshift of z = 6.295. Nature (2006) 1.70

Culture duration and conditions affect the oscillations of cytoplasmic calcium concentration induced by glucose in mouse pancreatic islets. Diabetologia (1994) 1.66

Influence of membrane potential changes on cytoplasmic Ca2+ concentration in an electrically excitable cell, the insulin-secreting pancreatic B-cell. J Biol Chem (1992) 1.64

Interplay between cytoplasmic Ca2+ and the ATP/ADP ratio: a feedback control mechanism in mouse pancreatic islets. Biochem J (1998) 1.59

Mechanisms by which glucose can control insulin release independently from its action on adenosine triphosphate-sensitive K+ channels in mouse B cells. J Clin Invest (1993) 1.59

Measurement of anti-DNA antibodies: a reappraisal using five different methods. Ann Rheum Dis (1987) 1.53

Hyperglycaemic effect of nifedipine. Br Med J (Clin Res Ed) (1981) 1.50

Phentolamine and yohimbine inhibit ATP-sensitive K+ channels in mouse pancreatic beta-cells. Br J Pharmacol (1990) 1.45

Mechanisms of the stimulation of insulin release by saturated fatty acids. A study of palmitate effects in mouse beta-cells. Diabetes (1994) 1.44

Tight links between adenine and guanine nucleotide pools in mouse pancreatic islets: a study with mycophenolic acid. Biochem J (1997) 1.43

Hierarchy of the beta-cell signals controlling insulin secretion. Eur J Clin Invest (2003) 1.39

The changes in adenine nucleotides measured in glucose-stimulated rodent islets occur in beta cells but not in alpha cells and are also observed in human islets. J Biol Chem (1998) 1.39

Neither adrenergic nor cholinergic antagonists in the central nervous system affect 2-deoxy-D-glucose(2-DG)-induced hyperglycemia. Brain Res (1990) 1.39

Tolbutamide stimulation and inhibition of insulin release: studies of the underlying ionic mechanisms in isolated rat islets. Diabetologia (1980) 1.34

Uptake and release of Ca2+ by the endoplasmic reticulum contribute to the oscillations of the cytosolic Ca2+ concentration triggered by Ca2+ influx in the electrically excitable pancreatic B-cell. J Biol Chem (1999) 1.33

Pronase effect on pancreatic beta cell secretion and morphology. Science (1973) 1.31

Insulin release independent of a rise in cytosolic free Ca2+ by forskolin and phorbol ester. FEBS Lett (1985) 1.27

The ionic, electrical, and secretory effects of endogenous cyclic adenosine monophosphate in mouse pancreatic B cells: studies with forskolin. Endocrinology (1984) 1.23

Influence of cell number on the characteristics and synchrony of Ca2+ oscillations in clusters of mouse pancreatic islet cells. J Physiol (1999) 1.22

Possible links between glucose-induced changes in the energy state of pancreatic B cells and insulin release. Unmasking by decreasing a stable pool of adenine nucleotides in mouse islets. J Clin Invest (1995) 1.21

Plasma endotoxin and serum cytokine levels in patients with alcoholic hepatitis: relation to severity of liver disturbance. Alcohol Clin Exp Res (2000) 1.20

Concentration dependence and time course of the effects of glucose on adenine and guanine nucleotides in mouse pancreatic islets. J Biol Chem (1996) 1.20

Effects of amino acids on membrane potential and 86Rb+ fluxes in pancreatic beta-cells. Am J Physiol (1981) 1.19

Who will care? Employment participation and willingness to supply informal care. J Health Econ (2009) 1.19

Surgical decompression of branch retinal vein occlusions. Arch Ophthalmol (1988) 1.18

Stable and diffusible pools of nucleotides in pancreatic islet cells. Endocrinology (1996) 1.17

Effects of putative activators of K+ channels in mouse pancreatic beta-cells. Br J Pharmacol (1989) 1.17

Cobalt inhibition of insulin secretion and calcium uptake by isolated rat islets. Am J Physiol (1975) 1.17

Cyclic variations of glucose-induced electrical activity in pancreatic B cells. Pflugers Arch (1982) 1.17

Tetraethylammonium potentiation of insulin release and inhibition of rubidium efflux in pancreatic islets. Biochem Biophys Res Commun (1977) 1.17

Intravitreal bevacizumab (Avastin) causing acute glaucoma: an unreported complication. Eye (Lond) (2007) 1.13

High incidence of hypoglycaemia in African patients treated with intravenous quinine for severe malaria. Br Med J (Clin Res Ed) (1987) 1.11

High glucose stimulates early response gene c-Myc expression in rat pancreatic beta cells. J Biol Chem (2001) 1.11

Imidazoline antagonists of alpha 2-adrenoceptors increase insulin release in vitro by inhibiting ATP-sensitive K+ channels in pancreatic beta-cells. Br J Pharmacol (1992) 1.11

The ionic, electrical, and secretory effects of protein kinase C activation in mouse pancreatic B-cells: studies with a phorbol ester. Endocrinology (1987) 1.10

Emptying of intracellular Ca2+ stores stimulates Ca2+ entry in mouse pancreatic beta-cells by both direct and indirect mechanisms. J Physiol (1997) 1.10

Quinine-induced modifications of insulin release and glucose metabolism by isolated pancreatic islets. FEBS Lett (1975) 1.10

Measurements of cytoplasmic Ca2+ in islet cell clusters show that glucose rapidly recruits beta-cells and gradually increases the individual cell response. Diabetes (2001) 1.10

Shortcomings of current models of glucose-induced insulin secretion. Diabetes Obes Metab (2009) 1.09

Children and car seats. Pediatrics (1986) 1.09

Hardening and termination of long-duration γ rays detected prior to lightning. Phys Rev Lett (2013) 1.08

Metabolic control of potassium permeability in pancreatic islet cells. Biochem J (1980) 1.07

Pulsatility of insulin and glucagon release: physiological significance and pharmacological implications. Diabetologia (1987) 1.07

Experimental ocular siderosis in the squirrel monkey. Am J Ophthalmol (1972) 1.06

The influence of gamma-aminobutyric acid on hormone release by the mouse and rat endocrine pancreas. Endocrinology (1991) 1.06

The labour market costs of community care. J Health Econ (1998) 1.05

Potassium dependence of the membrane potential of pancreatic B-cells. FEBS Lett (1978) 1.05

Glucagon immunoassay using polyethylene glycol to precipitate antibody-bound hormone. Diabetologia (1974) 1.04

Cell populations in the endocrine pancreas of human neonates and infants. Diabetologia (1981) 1.04

Disorganization of cytoplasmic Ca(2+) oscillations and pulsatile insulin secretion in islets from ob/ obmice. Diabetologia (2002) 1.03

Diet- and diabetes-induced changes of ob gene expression in rat adipose tissue. FEBS Lett (1995) 1.03

Distinct effects of glucose on the synchronous oscillations of insulin release and cytoplasmic Ca2+ concentration measured simultaneously in single mouse islets. Endocrinology (1995) 1.03

Phlorizin treatment of diabetic rats partially reverses the abnormal expression of genes involved in hepatic glucose metabolism. Diabetologia (1993) 1.02

Quinine and the stimulus-secretion coupling in pancreatic beta-cells: glucose-like effects on potassium permeability and insulin release. Endocrinology (1982) 1.02

The muscarinic receptor subtype in mouse pancreatic B-cells. FEBS Lett (1988) 1.01

The islet in type 2 diabetes: back to center stage. Diabetes (2001) 1.01

Temporal and quantitative correlations between insulin secretion and stably elevated or oscillatory cytoplasmic Ca2+ in mouse pancreatic beta-cells. Diabetes (1998) 1.01

Two sites of glucose control of insulin release with distinct dependence on the energy state in pancreatic B-cells. Biochem J (1994) 1.01

Muscarinic control of pancreatic B cell function involves sodium-dependent depolarization and calcium influx. Endocrinology (1988) 1.00

Oscillations of insulin secretion can be triggered by imposed oscillations of cytoplasmic Ca2+ or metabolism in normal mouse islets. Diabetes (1999) 1.00

The K+-ATP channel-independent pathway of regulation of insulin secretion by glucose: in search of the underlying mechanism. Diabetes (1998) 0.99

Anterior segment ischaemia following segmental scleral buckling. Br J Ophthalmol (1994) 0.99

Mechanism of the stimulation of insulin release in vitro by HB 699, a benzoic acid derivative similar to the non-sulphonylurea moiety of glibenclamide. Diabetologia (1985) 0.98

Effects of trifluoperazine and pimozide on stimulus-secretion coupling in pancreatic B-cells. Suggestion for a role of calmodulin? Biochem J (1981) 0.98

Intravenous amiodarone in the treatment of various arrhythmias following cardiac operations. J Thorac Cardiovasc Surg (1981) 0.97

The role of protein kinase-C in signal transduction through vasopressin and acetylcholine receptors in pancreatic B-cells from normal mouse. Endocrinology (1994) 0.97

A single mechanism for the stimulation of insulin release and 86Rb+ efflux from rat islets by cationic amino acids. Biochem J (1982) 0.97

Discovery of the short gamma-ray burst GRB 050709. Nature (2005) 0.96

Altered cAMP and Ca2+ signaling in mouse pancreatic islets with glucagon-like peptide-1 receptor null phenotype. Diabetes (1999) 0.96

Forskolin, an activator of adenylate cyclase, increases CA2+-dependent electrical activity induced by glucose in mouse pancreatic B cells. Endocrinology (1983) 0.96

Haeme-oxygenase 1 expression in rat pancreatic beta cells is stimulated by supraphysiological glucose concentrations and by cyclic AMP. Diabetologia (2003) 0.95

Dibutyryl cyclic AMP triggers Ca2+ influx and Ca2+-dependent electrical activity in pancreatic B cells. Biochem Biophys Res Commun (1983) 0.95

Increase in insulin release from rat pancreatic islets by quinolone antibiotics. Br J Pharmacol (1996) 0.95

Distinct mechanisms for two amplification systems of insulin release. Biochem J (1987) 0.95

Bicarbonate modulation of glucose-9nduced biphasic insulin release by rat islets. Am J Physiol (1976) 0.95

9-Aminoacridine- and tetraethylammonium-induced reduction of the potassium permeability in pancreatic B-cells. Effects on insulin release and electrical properties. Biochim Biophys Acta (1979) 0.94

Glucose-, calcium- and concentration-dependence of acetylcholine stimulation of insulin release and ionic fluxes in mouse islets. Biochem J (1988) 0.94

The potassium permeability of pancreatic islet cells: mechanisms of control and influence on insulin release. Horm Metab Res Suppl (1980) 0.94

Distinct effects of acetylcholine and glucose on 45calcium and 86rubidium efflux from mouse pancreatic islets. FEBS Lett (1984) 0.93

Trace elements in soils fertilized with poultry litter. Poult Sci (1999) 0.93

Children as passengers in automobiles: the neglected minority on the nation's highways. Pediatrics (1975) 0.93

Highly potent and stereoselective effects of the benzoic acid derivative AZ-DF 265 on pancreatic beta-cells. Br J Pharmacol (1988) 0.93

Increased glucose sensitivity of both triggering and amplifying pathways of insulin secretion in rat islets cultured for 1 wk in high glucose. Am J Physiol Endocrinol Metab (2004) 0.93