Published in Pharm Weekbl Sci on October 22, 1982
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Interaction of amiloride and its analogues with adenosine A1 receptors in calf brain. Biochem Pharmacol (1990) 0.82
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Quantification of the in vivo potency of the adenosine A2 receptor antagonist 8-(3-chlorostyryl)caffeine. J Pharmacol Exp Ther (1995) 0.82
Deoxyribose analogues of N6-cyclopentyladenosine (CPA): partial agonists at the adenosine A1 receptor in vivo. Br J Pharmacol (1995) 0.81
Novel competitive antagonists for P2 purinoceptors. Eur J Pharmacol (1994) 0.81
Relationships between structure and alpha-adrenergic receptor affinity of clonidine and some related cyclic amidines. Eur J Pharmacol (1981) 0.81
Pharmacokinetic-pharmacodynamic modelling of the cardiovascular effects of R- and S-N6-phenylisopropyladenosine in conscious normotensive rats. J Pharmacol Exp Ther (1995) 0.80
Distribution, excretion and metabolism of neuroleptics of the butyrophenone type. I. Excretion and metabolism of haloperidol and nine related butyrophenone-derivatives in the Wistar rat. Eur J Pharmacol (1967) 0.80
Mapping the xanthine C8-region of the adenosine A1 receptor with computer graphics. Eur J Pharmacol (1991) 0.79
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Pharmacokinetic-haemodynamic relationships of 2-chloroadenosine at adenosine A1 and A2a receptors in vivo. Br J Pharmacol (1996) 0.79
The mode of interaction of amiloride and some of its analogues with the adenosine A1 receptor. Neurochem Int (1992) 0.78
Nucleoside transport inhibition and platelet aggregation in human blood: R75231 and its enantiomers, draflazine and R88016. Eur J Pharmacol (1994) 0.78
The metabolism and excretion of cinnarizine by rats. Life Sci (1968) 0.78
Purification and characterization of enkephalin-degradating enzymes from calf-brain striatum. Biochem Biophys Res Commun (1983) 0.77
Structure-affinity relationship studies on 5-HT1A receptor ligands. 2. Heterobicyclic phenylpiperazines with N4-aralkyl substituents. J Med Chem (1994) 0.77
Localization of ( 3 H)pimozide in the rat brain in relation to its anti-amphetamine potency. J Pharm Pharmacol (1972) 0.77
Hybrid cholecystokinin-A antagonists based on molecular modeling of lorglumide and L-364,718. J Med Chem (1992) 0.76
Halopemide, a new psychotropic agent. Cerebral distribution and receptor interactions. Pharm Weekbl Sci (1985) 0.76
Effects of halopemide on GABA receptor binding, uptake and release. Brain Res (1981) 0.76
Opiate receptor interaction of compounds derived from or structurally related to fentanyl. J Med Chem (1981) 0.75
Regional localization of halopemide, a new psychotropic agent, in the rat brain. Eur J Pharmacol (1978) 0.75
Effect of various enkephalin analogs and dipeptides on the enzymatic activity of enkephalinase B isolated from calf-brain striatum. Life Sci (1986) 0.75
Distribution excretion and metabolism of neuroleptics of the butyrophenone type. II. Distribution, excretion and metabolism of haloperidol in Sprague-Dawley rats. Eur J Pharmacol (1967) 0.75
Research in the Division of Medicinal Chemistry. Pharm Weekbl Sci (1985) 0.75
Adenosine-A1 receptors are not coupled to Ca2+ uptake in rat brain synaptosomes. Biochem Pharmacol (1989) 0.75
Partial agonism of the nonselective adenosine receptor agonist 8-butylaminoadenosine at the A1 receptor in vivo. J Pharmacol Exp Ther (1996) 0.75
[3H]batrachotoxinin-A 20-alpha-benzoate binding to sodium channels in rat brain: sensitivity to tetrodotoxin and divalent cations. Eur J Pharmacol (1988) 0.75
Difenoxine (R15403), the active metabolite of diphenoxylate (R1132). 1. The excretion and metabolism in rats of difenoxine, the pharmacologically active metabolite of the antidiarrheal agent diphenoxylate. Arzneimittelforschung (1972) 0.75
Opiate receptor binding of nicomorphine and its hydrolysis products in rat brain. Eur J Pharmacol (1982) 0.75
A series of N4-imidoethyl derivatives of 1-(2,3-dihydro-1,4-benzodioxin-5-yl)piperazine as 5-HT1A receptor ligands: synthesis and structure-affinity relationships. J Med Chem (1995) 0.75
Effects of halopemide on potassium-induced release of radiolabeled neurotransmitters from rat cerebrocortical slices in vitro. Arch Int Pharmacodyn Ther (1980) 0.75
Effects of halopemide, a new psychotropic agent, on the uptake of serotonin by blood platelets. Arch Int Pharmacodyn Ther (1979) 0.75
Molecular modelling of asperlicin derived cholecystokinin A receptor antagonists. Eur J Pharmacol (1992) 0.75
Structure-affinity relationship studies on 5-HT1A receptor ligands. 1. Heterobicyclic phenylpiperazines with N4-alkyl substituents. J Med Chem (1993) 0.75
Isolation and characterization of an enkephalin-hydrolyzing dipeptidyl-aminopeptidase from calf-brain striatum. Neuropeptides (1985) 0.75
Molecular modelling of CCK-A receptors. Drug Des Discov (1994) 0.75
Regional distribution of halopemide, a new psychotropic agent, in the rat brain at different time intervals and after chronic administration. Life Sci (1979) 0.75
Peptides with a dual function: central neuroregulators and gut hormones. J Physiol (Paris) (1979) 0.75
Biotransformation of neuroleptanalgesics. Int Anesthesiol Clin (1974) 0.75
The metabolism and excretion of the neuroleptic drug pimozide (R 6238) by the wistar rat. Life Sci (1969) 0.75
The regional localization of R28935 in the cat brain as dependent on the route of administration. Naunyn Schmiedebergs Arch Pharmacol (1979) 0.75
Synthesis of enkephalinase B inhibitors, and their activity on isolated enkephalin-degrading enzymes. Eur J Pharmacol (1987) 0.75
The metabolism and excretion of benzetimide hydrochloride (R 4929) by rats. Life Sci (1968) 0.75
Computer modelling of the binding of non-selective ligands to biological receptors. Pharm Weekbl Sci (1983) 0.75
Inhibitors of calf-brain enkephalinase A and B. Life Sci (1983) 0.75
The regional localisation of a new potent centrally acting antihypertensive agent R 28935 and its less active threo-isomer R29814 in the cat brain. Eur J Pharmacol (1977) 0.75
Improved qualitative method for establishing flunitrazepam abuse using urine samples and column liquid chromatography with fluorimetric detection. J Chromatogr (1986) 0.75
Functional characteristics of a series of N4-substituted 1-(2,3-dihydro-1,4-benzodioxin-5-yl)piperazines as 5-HT1A receptor ligands. Structure-activity relationships. Bioorg Med Chem Lett (1998) 0.75
Halopemide and benzodiazepine binding sites. Arch Int Pharmacodyn Ther (1982) 0.75
The combined use of high-performance liquid chromatography and radioimmunoassay for the bioanalysis of nicomorphine and its metabolites. J Pharm Biomed Anal (1984) 0.75
Influence of the molecular structure of N6-(omega-aminoalkyl)adenosines on adenosine receptor affinity and intrinsic activity. Eur J Pharmacol (1989) 0.75