Synthesis of thiophene-2-carboxamidines containing 2-aminothiazoles and their biological evaluation as urokinase inhibitors.

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Published in Bioorg Med Chem Lett on April 09, 2001

Authors

K J Wilson1, C R Illig, N Subasinghe, J B Hoffman, M J Rudolph, R Soll, C J Molloy, R Bone, D Green, T Randall, M Zhang, F A Lewandowski, Z Zhou, C Sharp, D Maguire, B Grasberger, R L DesJarlais, J Spurlino

Author Affiliations

1: 3-Dimensional Pharmaceuticals, Inc., Exton, PA 19341, USA. wilson@3dp.com

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