PubRank

Patrick Dallemagne

Author PubWeight™ 7.37‹?›

Top papers

Rank Title Journal Year PubWeight™‹?›
1 Synthesis and preliminary in vitro evaluation of antimycobacterial activity of new pyrrolo[1,2-a] quinoxaline-carboxylic acid hydrazide derivatives. J Enzyme Inhib Med Chem 2004 0.95
2 Synthesis of a novel class of non-peptide NK-2 receptor ligand, derived from 1-phenyl-3-pyrrol-1-ylindan-2-carboxamides. Bioorg Med Chem 2002 0.92
3 Synergistic effect of acetylcholinesterase inhibition (donepezil) and 5-HT(4) receptor activation (RS67333) on object recognition in mice. Behav Brain Res 2012 0.84
4 MR22388, a novel anti-cancer agent with a strong FLT-3 ITD kinase affinity. Cancer Lett 2012 0.80
5 Synthesis of new 4-[2-(alkylamino) ethylthio]pyrrolo[1,2-a]quinoxaline and 5-[2-(alkylamino) ethylthio]pyrrolo[1,2-a]thieno[3,2-e]pyrazine derivatives, as potential bacterial multidrug resistance pump inhibitors. J Enzyme Inhib Med Chem 2007 0.80
6 Hydrogenative desulphurization of thienopyrrolizinones: an easy and selective access to (Z)-phenethylidenepyrrolizinones with in vitro cytotoxic activity. Eur J Med Chem 2009 0.78
7 Tripentones: a promising series of potent anti-cancer agents. Anticancer Agents Med Chem 2009 0.77
8 Synthesis and biological evaluation of thienopyrrolizines, a new family of CDK/GSK-3 inhibitors. J Enzyme Inhib Med Chem 2004 0.77
9 Synthesis, antimalarial activity, and molecular modeling of new pyrrolo[1,2-a]quinoxalines, bispyrrolo[1,2-a]quinoxalines, bispyrido[3,2-e]pyrrolo[1,2-a]pyrazines, and bispyrrolo[1,2-a]thieno[3,2-e]pyrazines. J Med Chem 2004 0.76
10 Virtual screening discovery of new acetylcholinesterase inhibitors issued from CERMN chemical library. J Chem Inf Model 2010 0.76
11 A first cyclopenta[c]thiophene dimer as a new bivalent potent cytotoxic derivative. J Enzyme Inhib Med Chem 2002 0.75
12 Synthesis of novel 7-oxo and 7-hydroxy trifluoroallocolchicinoids with cytotoxic effect. Bioorg Med Chem 2012 0.75
13 Synthesis and preliminary in vivo evaluation of new 2-Aryl-6-methyl-1,2-dihydro-1H-pyridin-4-ones and 2-Aryl-6-methylpiperidin-4-ols, as potential anti-amnesiant agents. J Enzyme Inhib Med Chem 2005 0.75
14 Synthesis and biological evaluation of new donepezil-like Thiaindanones as AChE inhibitors. J Enzyme Inhib Med Chem 2008 0.75
15 N-substituted piperazinopyridylsteroid derivatives as abiraterone analogues inhibit growth and induce pro-apoptosis in human hormone-independent prostate cancer cell lines. Chem Biol Drug Des 2013 0.75
16 Synthesis, reactivity and biological evaluation of novel halogenated tripentones. Bioorg Med Chem 2009 0.75
17 Synthesis and initial results for MAO-B inhibition by new N-propargyl-3-pyrrol-1-ylindanamine derivatives, analogues of rasagiline. J Enzyme Inhib Med Chem 2003 0.75
18 Synthesis of new bisaryl cyclopentathiophene and thienocyclopentoxazolidine derivatives as potential cytotoxic agents. J Enzyme Inhib Med Chem 2007 0.75
19 Intramolecular cyclisation of β-aryl-β-amino acids in the design of novel heterocyclic systems with therapeutic interest: an unfailing source of diversity. Curr Med Chem 2010 0.75
20 Synthesis of new dipyrrolo- and furopyrrolopyrazinones related to tripentones and their biological evaluation as potential kinases (CDKs1-5, GSK-3) inhibitors. Eur J Med Chem 2008 0.75
21 [Study of in vitro cytotoxic activity of cyclopentanones derivatives]. Tunis Med 2004 0.75
22 Synthesis and biological evaluation as AChE inhibitors of new indanones and thiaindanones related to donepezil. Eur J Med Chem 2005 0.75