Published in J Org Chem on June 25, 2004
Novel 2-[(benzylamino)methyl]pyrrolidine-3,4-diol derivatives as alpha-mannosidase inhibitors and with antitumor activities against hematological and solid malignancies. Bioorg Med Chem (2010) 1.40
Rational design of indoleamine 2,3-dioxygenase inhibitors. J Med Chem (2010) 1.22
Organosulfur compounds: electrophilic reagents in transition-metal-catalyzed carbon-carbon bond-forming reactions. Angew Chem Int Ed Engl (2005) 0.99
Recent synthetic approaches toward non-anomeric spiroketals in natural products. Molecules (2008) 0.97
Silyl methallylsulfinates: efficient and powerful agents for the chemoselective silylation of alcohols, polyols, phenols and carboxylic acids. Chem Commun (Camb) (2005) 0.93
Structural insights into the specificity of Xyn10B from Paenibacillus barcinonensis and its improved stability by forced protein evolution. J Biol Chem (2009) 0.91
Synthesis of the C(1)-C(11) polyene fragment of apoptolidin with a new sulfur dioxide-based organic chemistry. Chemistry (2005) 0.90
Synthesis of novel pyrrolidine 3,4-diol derivatives as inhibitors of alpha-L-fucosidases. Org Biomol Chem (2009) 0.85
New efficient route to an advanced precursor of the AB spiroketal of spongistatins. Org Lett (2007) 0.85
Rational design of 4-aryl-1,2,3-triazoles for indoleamine 2,3-dioxygenase 1 inhibition. J Med Chem (2012) 0.85
Parallel solution-phase and microwave-assisted synthesis of new S-DABO derivatives endowed with subnanomolar anti-HIV-1 activity. J Med Chem (2005) 0.85
Scope and limitations of the double [4+3]-cycloadditions of 2-oxyallyl cations to 2,2'-methylenedifuran and derivatives. J Org Chem (2003) 0.84
New synthetic seven-membered 1-azasugars displaying potent inhibition towards glycosidases and glucosylceramide transferase. Chembiochem (2008) 0.84
Discovery, molecular and pharmacological characterization of GSA-10, a novel small-molecule positive modulator of Smoothened. Mol Pharmacol (2013) 0.84
Short synthesis of the C16-C28 polyketide fragment of apoptolidin A aglycone. Chem Commun (Camb) (2007) 0.83
Palladium-catalyzed Stille cross-couplings of sulfonyl chlorides and organostannanes. J Am Chem Soc (2003) 0.82
Total synthesis and determination of the absolute configuration of (-)-dolabriferol. Angew Chem Int Ed Engl (2010) 0.82
New concise total synthesis of (+)-lentiginosine and some structural analogues. J Org Chem (2005) 0.81
Microwave-assisted intramolecular Huisgen cycloaddition of azido alkynes derived from alpha-amino acids. J Org Chem (2009) 0.81
Synthesis and conformational analysis of (alpha-D-galactosyl)phenylmethane and alpha-,beta-difluoromethane analogues: interactions with the plant lectin viscumin. Chemistry (2009) 0.81
Synthesis and anti-HIV activity of trivalent CD4-mimetic miniproteins. Bioorg Med Chem (2007) 0.80
Microwave-assisted aminocarbonylation of ynamides by using catalytic [Fe3(CO)12] at low pressures of carbon monoxide. Chemistry (2011) 0.80
Functionalized pyrrolidines inhibit alpha-mannosidase activity and growth of human glioblastoma and melanoma cells. J Med Chem (2005) 0.80
Glycosidase inhibitors as potential HIV entry inhibitors? Curr Drug Metab (2004) 0.79
Iron-catalyzed desulfinylative C-C cross-coupling reactions of sulfonyl chlorides with grignard reagents. Angew Chem Int Ed Engl (2008) 0.79
Palladium-catalyzed Suzuki-Miyaura cross-couplings of sulfonyl chlorides and boronic acids. Org Lett (2004) 0.79
Search for alpha-glucosidase inhibitors: new N-substituted valienamine and conduramine F-1 derivatives. Bioorg Med Chem (2006) 0.79
Tandem Staudinger-azaWittig mediated ring expansion: rapid access to new isofagomine-tetrahydroxyazepane hybrids. Chem Commun (Camb) (2006) 0.79
A C-linked disaccharide analogue of Thomsen-Friedenreich epitope induces a strong immune response in mice. Chemistry (2012) 0.78
Stereoselective syntheses of 1,4-dideoxy-1,4-imino-octitols and novel tetrahydroxyindolizidines. J Org Chem (2003) 0.78
Chemoselective C-H bond activation: ligand and solvent free iron-catalyzed oxidative C-C cross-coupling of tertiary amines with terminal alkynes. Reaction scope and mechanism. Org Lett (2009) 0.78
6-Azido hyacinthacine A2 gives a straightforward access to the first multivalent pyrrolizidine architectures. Org Biomol Chem (2014) 0.78
Nucleophilic opening of epoxyazepanes: expanding the family of polyhydroxyazepane-based glycosidase inhibitors. Org Biomol Chem (2006) 0.78
An efficient combinatorial method for the discovery of glycosidase inhibitors. Chembiochem (2002) 0.78
Design and synthesis of acetamido tri- and tetra-hydroxyazepanes: potent and selective beta-N-acetylhexosaminidase inhibitors. Bioorg Med Chem (2009) 0.78
Total asymmetric synthesis of (-)-conduramine B-1 and of its enantiomer. N-Benzyl derivatives of conduramine B-1 are beta-glucosidase inhibitors. Bioorg Med Chem Lett (2005) 0.78
Synthesis of (E,Z)-1-alkoxy-3-acyloxy-2-methylpenta-1,3-dienes via Danishefsky-type dienes or O-acylation of enones. J Org Chem (2009) 0.77
Ab initio and experimental studies on the hetero-Diels-Alder and cheletropic additions of sulfur dioxide to (E)-1-methoxybutadiene: a mechanism involving three molecules of SO(2). J Org Chem (2002) 0.77
Synthesis of new oxathiazinane dioxides and their in vitro cancer cell growth inhibitory activity. Bioorg Med Chem Lett (2009) 0.77
The first synthesis of substituted azepanes mimicking monosaccharides: a new class of potent glycosidase inhibitors. Org Biomol Chem (2004) 0.77
Desulfinylation of prop-2-enesulfinic acid: experimental results and mechanistic theoretical analysis. J Am Chem Soc (2009) 0.77
Synthesis of optically active 5-alkoxy-6-methylcyclohex-2-en-1-ones and 4-alkoxy-5-methylcyclopent-1-enyl benzoate. J Org Chem (2009) 0.77
Sulfur dioxide mediated one-pot, three- and four-component syntheses of polyfunctional sulfonamides and sulfonic esters: study of the stereoselectivity of the ene reaction of sulfur dioxide. J Org Chem (2004) 0.77
A multidisciplinary approach for the identification of novel HIV-1 non-nucleoside reverse transcriptase inhibitors: S-DABOCs and DAVPs. ChemMedChem (2008) 0.77
The anti-lymphoma activity of APO866, an inhibitor of nicotinamide adenine dinucleotide biosynthesis, is potentialized when used in combination with anti-CD20 antibody. Leuk Lymphoma (2014) 0.76
Anti-cancer activity of 5-O-alkyl 1,4-imino-1,4-dideoxyribitols. Bioorg Med Chem (2011) 0.76
An improved synthesis of alpha,beta-unsaturated nitrones relevant to the stephacidins and analogs thereof. Bioorg Med Chem Lett (2009) 0.76
Three dimensional structure of a bacterial α-l-fucosidase with a 5-membered iminocyclitol inhibitor. Bioorg Med Chem (2013) 0.76
Parallel solution-phase synthesis of 4-dialkylamino-2-methylsulfonyl-6-vinylpyrimidines. J Comb Chem (2005) 0.76
Effects of ethylene glycol addition on the aggregation and micellar growth of gemini surfactants. Langmuir (2006) 0.76
Amine-linked diglycosides: Synthesis facilitated by the enhanced reactivity of allylic electrophiles, and glycosidase inhibition assays. Beilstein J Org Chem (2011) 0.76
Specific activation of ERK pathways by chitin oligosaccharides in embryonic zebrafish cell lines. Glycobiology (2003) 0.76
Concise synthesis of complicated polypropionates through one-pot dissymmetrical two-directional chain elongation. Chemistry (2011) 0.76
Polysulfones: catalysts for alkene isomerization. Angew Chem Int Ed Engl (2004) 0.76
Total asymmetric syntheses of β-hydroxy-δ-lactones via Umpolung with sulfur dioxide. J Org Chem (2011) 0.75
Synthesis and physicochemical characterization of alkanedyil-α-ω-bis(dimethyldodecylammonium) bromide, 12-s-12,2Br-, surfactants with s=7, 9, 11 in aqueous medium. J Colloid Interface Sci (2012) 0.75
Synthesis, biological evaluation, WAC and NMR studies of S-galactosides and non-carbohydrate ligands of cholera toxin based on polyhydroxyalkylfuroate moieties. Chemistry (2013) 0.75
Synthesis of long-chain polyketide fragments by reaction of 1,3-dioxy-1,3-dienes with allylsilanes: umpolung with sulfur dioxide. Org Lett (2004) 0.75
Physicochemical characterization of bromide mono- and dimeric surfactants with phenyl and cyclohexyl rings in the head group. J Colloid Interface Sci (2011) 0.75
Spirocyclopropyl pyrrolidines as a new series of alpha-L-fucosidase inhibitors. Bioorg Med Chem (2006) 0.75
Syntheses and biological activities of 1,4-iminoalditol derivatives as alpha-L-fucosidase inhibitors. Chimia (Aarau) (2011) 0.75
Allyl, methallyl, prenyl, and methylprenyl ethers as protected alcohols: their selective cleavage with diphenyldisulfone under neutral conditions. Org Lett (2004) 0.75
The catalyzed desulfinylative allylation of carbonyl compounds with alk-2-enesulfonyl chlorides and silyl alk-2-enesulfinates. Chemistry (2010) 0.75
Synthesis and glycosidase inhibitory activities of 2-(aminoalkyl)pyrrolidine-3,4-diol derivatives. Bioorg Med Chem (2003) 0.75
Combinatorial chemistry as a tool for targeting different stages of the replicative HIV-1 cycle. Comb Chem High Throughput Screen (2005) 0.75
Microwave-assisted carbonylation and cyclocarbonylation of aryl iodides under ligand free heterogeneous catalysis. J Org Chem (2010) 0.75
Synthesis of enantiomerically pure 1,2-diamine derivatives of 7-azabicyclo[2.2.1]heptane. New leads as glycosidase inhibitors and rigid scaffolds for the preparation of peptide analogues. J Org Chem (2003) 0.75
Mechanism of the diphenyldisulfone-catalyzed isomerization of alkenes. Origin of the chemoselectivity: experimental and quantum chemistry studies. J Am Chem Soc (2006) 0.75
The spirocyclopropyl moiety as a methyl surrogate in the structure of l-fucosidase and l-rhamnosidase inhibitors. Bioorg Med Chem (2009) 0.75
First asymmetric synthesis of the cyclohexanone subunit of baconipyrones A and B. Revision of its structure. Org Lett (2004) 0.75
Synthesis of [(2S,3S,4R)-3,4-dihydroxypyrrolidin-2-yl]-5-methylfuran-4-carboxylic acid derivatives: new leads as selective beta-galactosidase inhibitors. Bioorg Med Chem Lett (2002) 0.75
Sulfur dioxide-mediated syntheses of polyfunctional alkenes and (E,Z)- and (E,E)-2,4-dien-1-ones. Org Lett (2005) 0.75
Equilibrium and kinetic deuterium isotope effects on the hetero-Diels-Alder addition of sulfur dioxide. Angew Chem Int Ed Engl (2003) 0.75
Expeditious asymmetric synthesis of a stereoheptad corresponding to the C(19)-C(27)-ansa chain of rifamycins: formal total synthesis of Rifamycin S. Chemistry (2005) 0.75
Polysulfones: solid organic catalysts for the chemoselective cleavage of methyl-substituted allyl ethers under neutral conditions. Chem Commun (Camb) (2004) 0.75
A short and convenient synthesis of 1-deoxymannojirimycin and N-oxy analogues from D-fructose. J Org Chem (2009) 0.75
The use of levoglucosenone and isolevoglucosenone as templates for the construction of C-linked disaccharides. Carbohydr Res (2006) 0.75
BCl3-mediated ene reaction of sulfur dioxide and unfunctionalized alkenes. Chemistry (2010) 0.75
Synthesis and conformational analysis of novel trimeric maleimide cross-linking reagents. J Org Chem (2007) 0.75
Short diastereoselective synthesis of the C1-C13 (AB spiroacetal) and C17-C28 fragments (CD spiroacetal) of spongistatin 1 and 2 through double chain-elongation reactions. Chemistry (2010) 0.75
Exploiting the ring strain in bicyclo[2.2.1]heptane systems for the stereoselective preparation of highly functionalized cyclopentene, dihydrofuran, pyrroline, and pyrrolidine scaffolds. Org Lett (2011) 0.75
Monosaccharides and analogues from simple achiral unsaturated compounds. Chimia (Aarau) (2011) 0.75
The norbornene mystery revealed. Chem Commun (Camb) (2010) 0.75
Synthesis and inhibitory activities of novel C-3 substituted azafagomines: a new type of selective inhibitors of α-L-fucosidases. Bioorg Med Chem (2010) 0.75
C-linked disaccharide analogue of the Thomsen-Friedenreich (T)-epitope alpha-O-conjugated to L-serine. Chemistry (2005) 0.75
Rapid discovery of potent α-fucosidase inhibitors by in situ screening of a library of (pyrrolidin-2-yl)triazoles. Org Biomol Chem (2014) 0.75
Synthesis and biological evaluation of 4-alkylamino-6-(2-hydroxyethyl)-2-methylthiopyrimidines as new rubella virus inhibitors. Eur J Med Chem (2006) 0.75
Synthesis and glycosidase inhibitory activity of 1-amino-3,6-anhydro-1-deoxy-D-sorbitol derivatives. Bioorg Chem (2009) 0.75
Strain-promoted retro-Dieckmann-type condensation on [2.2.2]- and [2.2.1]bicyclic systems: a fragmentation reaction for the preparation of functionalized heterocycles and carbocycles. Org Biomol Chem (2013) 0.75
Glycochemistry today. Chimia (Aarau) (2011) 0.75
Palladium-catalyzed conversion of beta,gamma-unsaturated silyl sulfinates into (E)-alkenes: asymmetric synthesis of polypropionate fragments. J Org Chem (2004) 0.75
Carbohydrates in sustainable development, Part 1. Renewable resources for chemistry and biotechnology. Preface. Top Curr Chem (2010) 0.75
Allenyl sulfones and allenyl sulfides in the synthesis of 3-pyrrolines. A novel nucleophilic [3 + 2] cycloaddition on allenyl sulfones giving rearranged cycloadducts. Org Lett (2009) 0.75