Published in Org Lett on January 08, 2004
Synthesis of aryl sulfonamides via palladium-catalyzed chlorosulfonylation of arylboronic acids. J Am Chem Soc (2013) 0.91
Novel 2-[(benzylamino)methyl]pyrrolidine-3,4-diol derivatives as alpha-mannosidase inhibitors and with antitumor activities against hematological and solid malignancies. Bioorg Med Chem (2010) 1.40
Rational design of indoleamine 2,3-dioxygenase inhibitors. J Med Chem (2010) 1.22
Organosulfur compounds: electrophilic reagents in transition-metal-catalyzed carbon-carbon bond-forming reactions. Angew Chem Int Ed Engl (2005) 0.99
Recent synthetic approaches toward non-anomeric spiroketals in natural products. Molecules (2008) 0.97
Silyl methallylsulfinates: efficient and powerful agents for the chemoselective silylation of alcohols, polyols, phenols and carboxylic acids. Chem Commun (Camb) (2005) 0.93
Structural insights into the specificity of Xyn10B from Paenibacillus barcinonensis and its improved stability by forced protein evolution. J Biol Chem (2009) 0.91
Synthesis of the C(1)-C(11) polyene fragment of apoptolidin with a new sulfur dioxide-based organic chemistry. Chemistry (2005) 0.90
Rational design of 4-aryl-1,2,3-triazoles for indoleamine 2,3-dioxygenase 1 inhibition. J Med Chem (2012) 0.85
New efficient route to an advanced precursor of the AB spiroketal of spongistatins. Org Lett (2007) 0.85
Synthesis of novel pyrrolidine 3,4-diol derivatives as inhibitors of alpha-L-fucosidases. Org Biomol Chem (2009) 0.85
New synthetic seven-membered 1-azasugars displaying potent inhibition towards glycosidases and glucosylceramide transferase. Chembiochem (2008) 0.84
Scope and limitations of the double [4+3]-cycloadditions of 2-oxyallyl cations to 2,2'-methylenedifuran and derivatives. J Org Chem (2003) 0.84
Short synthesis of the C16-C28 polyketide fragment of apoptolidin A aglycone. Chem Commun (Camb) (2007) 0.83
Total synthesis and determination of the absolute configuration of (-)-dolabriferol. Angew Chem Int Ed Engl (2010) 0.82
Palladium-catalyzed Stille cross-couplings of sulfonyl chlorides and organostannanes. J Am Chem Soc (2003) 0.82
Synthesis and conformational analysis of (alpha-D-galactosyl)phenylmethane and alpha-,beta-difluoromethane analogues: interactions with the plant lectin viscumin. Chemistry (2009) 0.81
New concise total synthesis of (+)-lentiginosine and some structural analogues. J Org Chem (2005) 0.81
Functionalized pyrrolidines inhibit alpha-mannosidase activity and growth of human glioblastoma and melanoma cells. J Med Chem (2005) 0.80
Glycosidase inhibitors as potential HIV entry inhibitors? Curr Drug Metab (2004) 0.79
Search for alpha-glucosidase inhibitors: new N-substituted valienamine and conduramine F-1 derivatives. Bioorg Med Chem (2006) 0.79
Tandem Staudinger-azaWittig mediated ring expansion: rapid access to new isofagomine-tetrahydroxyazepane hybrids. Chem Commun (Camb) (2006) 0.79
Iron-catalyzed desulfinylative C-C cross-coupling reactions of sulfonyl chlorides with grignard reagents. Angew Chem Int Ed Engl (2008) 0.79
A C-linked disaccharide analogue of Thomsen-Friedenreich epitope induces a strong immune response in mice. Chemistry (2012) 0.78
Stereoselective syntheses of 1,4-dideoxy-1,4-imino-octitols and novel tetrahydroxyindolizidines. J Org Chem (2003) 0.78
Chemoselective C-H bond activation: ligand and solvent free iron-catalyzed oxidative C-C cross-coupling of tertiary amines with terminal alkynes. Reaction scope and mechanism. Org Lett (2009) 0.78
Nucleophilic opening of epoxyazepanes: expanding the family of polyhydroxyazepane-based glycosidase inhibitors. Org Biomol Chem (2006) 0.78
An efficient combinatorial method for the discovery of glycosidase inhibitors. Chembiochem (2002) 0.78
Design and synthesis of acetamido tri- and tetra-hydroxyazepanes: potent and selective beta-N-acetylhexosaminidase inhibitors. Bioorg Med Chem (2009) 0.78
Total asymmetric synthesis of (-)-conduramine B-1 and of its enantiomer. N-Benzyl derivatives of conduramine B-1 are beta-glucosidase inhibitors. Bioorg Med Chem Lett (2005) 0.78
Synthesis of optically active 5-alkoxy-6-methylcyclohex-2-en-1-ones and 4-alkoxy-5-methylcyclopent-1-enyl benzoate. J Org Chem (2009) 0.77
Desulfinylation of prop-2-enesulfinic acid: experimental results and mechanistic theoretical analysis. J Am Chem Soc (2009) 0.77
Synthesis of (E,Z)-1-alkoxy-3-acyloxy-2-methylpenta-1,3-dienes via Danishefsky-type dienes or O-acylation of enones. J Org Chem (2009) 0.77
Sulfur dioxide mediated one-pot, three- and four-component syntheses of polyfunctional sulfonamides and sulfonic esters: study of the stereoselectivity of the ene reaction of sulfur dioxide. J Org Chem (2004) 0.77
Synthesis of new oxathiazinane dioxides and their in vitro cancer cell growth inhibitory activity. Bioorg Med Chem Lett (2009) 0.77
The first synthesis of substituted azepanes mimicking monosaccharides: a new class of potent glycosidase inhibitors. Org Biomol Chem (2004) 0.77
Ab initio and experimental studies on the hetero-Diels-Alder and cheletropic additions of sulfur dioxide to (E)-1-methoxybutadiene: a mechanism involving three molecules of SO(2). J Org Chem (2002) 0.77
Anti-cancer activity of 5-O-alkyl 1,4-imino-1,4-dideoxyribitols. Bioorg Med Chem (2011) 0.76
Concise synthesis of complicated polypropionates through one-pot dissymmetrical two-directional chain elongation. Chemistry (2011) 0.76
Polysulfones: catalysts for alkene isomerization. Angew Chem Int Ed Engl (2004) 0.76
The anti-lymphoma activity of APO866, an inhibitor of nicotinamide adenine dinucleotide biosynthesis, is potentialized when used in combination with anti-CD20 antibody. Leuk Lymphoma (2014) 0.76
Total asymmetric syntheses of β-hydroxy-δ-lactones via Umpolung with sulfur dioxide. J Org Chem (2011) 0.75
Carbohydrates in sustainable development, Part 1. Renewable resources for chemistry and biotechnology. Preface. Top Curr Chem (2010) 0.75
Synthesis of long-chain polyketide fragments by reaction of 1,3-dioxy-1,3-dienes with allylsilanes: umpolung with sulfur dioxide. Org Lett (2004) 0.75
Palladium-catalyzed conversion of beta,gamma-unsaturated silyl sulfinates into (E)-alkenes: asymmetric synthesis of polypropionate fragments. J Org Chem (2004) 0.75
Allyl, methallyl, prenyl, and methylprenyl ethers as protected alcohols: their selective cleavage with diphenyldisulfone under neutral conditions. Org Lett (2004) 0.75
The catalyzed desulfinylative allylation of carbonyl compounds with alk-2-enesulfonyl chlorides and silyl alk-2-enesulfinates. Chemistry (2010) 0.75
Synthesis of branched seven-membered 1-N-iminosugars and their evaluation as glycosidase inhibitors. Carbohydr Res (2011) 0.75
Synthesis and glycosidase inhibitory activities of 2-(aminoalkyl)pyrrolidine-3,4-diol derivatives. Bioorg Med Chem (2003) 0.75
Amide formation in one pot from carboxylic acids and amines via carboxyl and sulfinyl mixed anhydrides. Org Lett (2013) 0.75
The spirocyclopropyl moiety as a methyl surrogate in the structure of l-fucosidase and l-rhamnosidase inhibitors. Bioorg Med Chem (2009) 0.75
Synthesis of enantiomerically pure 1,2-diamine derivatives of 7-azabicyclo[2.2.1]heptane. New leads as glycosidase inhibitors and rigid scaffolds for the preparation of peptide analogues. J Org Chem (2003) 0.75
Mechanism of the diphenyldisulfone-catalyzed isomerization of alkenes. Origin of the chemoselectivity: experimental and quantum chemistry studies. J Am Chem Soc (2006) 0.75
Synthesis of d- and l-2,3-trans-3,4-cis-4,5-trans-3,4-dihydroxy-5-hydroxymethylproline and tripeptides containing them. J Org Chem (2004) 0.75
First asymmetric synthesis of the cyclohexanone subunit of baconipyrones A and B. Revision of its structure. Org Lett (2004) 0.75
Sulfur dioxide-mediated syntheses of polyfunctional alkenes and (E,Z)- and (E,E)-2,4-dien-1-ones. Org Lett (2005) 0.75
Amides in one pot from carboxylic acids and amines via sulfinylamides. Org Lett (2014) 0.75
Polysulfones: solid organic catalysts for the chemoselective cleavage of methyl-substituted allyl ethers under neutral conditions. Chem Commun (Camb) (2004) 0.75
The hetero-Diels-Alder addition of sulfur dioxide: the pseudo-chair conformation of a 4,5-dialkylsultine. Chemistry (2003) 0.75
Spirocyclopropyl pyrrolidines as a new series of alpha-L-fucosidase inhibitors. Bioorg Med Chem (2006) 0.75
A short and convenient synthesis of 1-deoxymannojirimycin and N-oxy analogues from D-fructose. J Org Chem (2009) 0.75
Stereoselective synthesis of (2S,3S,4R,5S)-5-methylpyrrolidine-3,4-diol derivatives that are highly selective alpha-L-fucosidase inhibitors. Chem Commun (Camb) (2005) 0.75
Synthesis of [(2S,3S,4R)-3,4-dihydroxypyrrolidin-2-yl]-5-methylfuran-4-carboxylic acid derivatives: new leads as selective beta-galactosidase inhibitors. Bioorg Med Chem Lett (2002) 0.75
Short diastereoselective synthesis of the C1-C13 (AB spiroacetal) and C17-C28 fragments (CD spiroacetal) of spongistatin 1 and 2 through double chain-elongation reactions. Chemistry (2010) 0.75
Equilibrium and kinetic deuterium isotope effects on the hetero-Diels-Alder addition of sulfur dioxide. Angew Chem Int Ed Engl (2003) 0.75
Expeditious asymmetric synthesis of a stereoheptad corresponding to the C(19)-C(27)-ansa chain of rifamycins: formal total synthesis of Rifamycin S. Chemistry (2005) 0.75
The norbornene mystery revealed. Chem Commun (Camb) (2010) 0.75
The use of levoglucosenone and isolevoglucosenone as templates for the construction of C-linked disaccharides. Carbohydr Res (2006) 0.75
BCl3-mediated ene reaction of sulfur dioxide and unfunctionalized alkenes. Chemistry (2010) 0.75
Synthesis and glycosidase inhibitory activity of 1-amino-3,6-anhydro-1-deoxy-D-sorbitol derivatives. Bioorg Chem (2009) 0.75
Glycochemistry today. Chimia (Aarau) (2011) 0.75
C-linked disaccharide analogue of the Thomsen-Friedenreich (T)-epitope alpha-O-conjugated to L-serine. Chemistry (2005) 0.75