Rank |
Title |
Journal |
Year |
PubWeight™‹?› |
1
|
Multidrug resistance reversal agents.
|
J Med Chem
|
2003
|
1.42
|
2
|
8-O-Azeloyl-14-benzoylaconine: a new alkaloid from the roots of Aconitum karacolicum Rapcs and its antiproliferative activities.
|
Bioorg Med Chem
|
2005
|
0.95
|
3
|
Synthesis and preliminary in vitro evaluation of antimycobacterial activity of new pyrrolo[1,2-a] quinoxaline-carboxylic acid hydrazide derivatives.
|
J Enzyme Inhib Med Chem
|
2004
|
0.95
|
4
|
Synthesis of new pyrrolo[1,2-a]quinoxaline derivatives as potential inhibitors of Akt kinase.
|
J Enzyme Inhib Med Chem
|
2008
|
0.93
|
5
|
Synthesis of a novel class of non-peptide NK-2 receptor ligand, derived from 1-phenyl-3-pyrrol-1-ylindan-2-carboxamides.
|
Bioorg Med Chem
|
2002
|
0.92
|
6
|
Probing the role of the covalent linkage of ferrocene into a chloroquine template.
|
J Med Chem
|
2006
|
0.87
|
7
|
Synthesis, analytical behaviour and biological evaluation of new 4-substituted pyrrolo[1,2-a]quinoxalines as antileishmanial agents.
|
Bioorg Med Chem
|
2006
|
0.86
|
8
|
Synthesis and preliminary evaluation of new 1- and 3-[1-(2-hydroxy-3-phenoxypropyl)]xanthines from 2-amino-2-oxazolines as potential A1 and A2A adenosine receptor antagonists.
|
Bioorg Med Chem
|
2005
|
0.81
|
9
|
Hemisynthesis and antiproliferative properties of mono-[O-(14-benzoylaconine-8-yl)]esters and bis-[O-(14-benzoylaconine-8-yl)]esters.
|
Eur J Med Chem
|
2012
|
0.81
|
10
|
Synthesis of new 4-[2-(alkylamino) ethylthio]pyrrolo[1,2-a]quinoxaline and 5-[2-(alkylamino) ethylthio]pyrrolo[1,2-a]thieno[3,2-e]pyrazine derivatives, as potential bacterial multidrug resistance pump inhibitors.
|
J Enzyme Inhib Med Chem
|
2007
|
0.80
|
11
|
Modulation of cell proliferation in rat liver cell cultures by new calix[4]arenes.
|
J Enzyme Inhib Med Chem
|
2006
|
0.79
|
12
|
Synthesis of omeprazole analogues and evaluation of these as potential inhibitors of the multidrug efflux pump NorA of Staphylococcus aureus.
|
Antimicrob Agents Chemother
|
2006
|
0.79
|
13
|
Synthesis and evaluation of the antiproliferative activity of novel pyrrolo[1,2-a]quinoxaline derivatives, potential inhibitors of Akt kinase. Part II.
|
J Enzyme Inhib Med Chem
|
2010
|
0.79
|
14
|
New ferrocenic pyrrolo[1,2-a]quinoxaline derivatives: synthesis, and in vitro antimalarial activity.
|
Bioorg Med Chem
|
2008
|
0.78
|
15
|
New ferrocenic pyrrolo[1,2-a]quinoxaline derivatives: synthesis, and in vitro antimalarial activity--Part II.
|
Eur J Med Chem
|
2011
|
0.77
|
16
|
Synthesis, antimalarial activity, and molecular modeling of new pyrrolo[1,2-a]quinoxalines, bispyrrolo[1,2-a]quinoxalines, bispyrido[3,2-e]pyrrolo[1,2-a]pyrazines, and bispyrrolo[1,2-a]thieno[3,2-e]pyrazines.
|
J Med Chem
|
2004
|
0.76
|
17
|
Antiproliferative effect on HepaRG cell cultures of new calix[4]arenes. Part II.
|
J Enzyme Inhib Med Chem
|
2010
|
0.76
|
18
|
Synthesis of new 4-(E)-alkenylpyrrolo[1,2-a]quinoxalines as antileishmanial agents by Suzuki-Miyaura cross-coupling reactions.
|
J Enzyme Inhib Med Chem
|
2007
|
0.75
|
19
|
Development of a rapid RP-HPLC method for the determination of clonazepam in human plasma.
|
J Pharm Biomed Anal
|
2004
|
0.75
|
20
|
Highly diastereoselective synthesis of C6-functionalized dihydroimidazotriazines.
|
Org Lett
|
2003
|
0.75
|
21
|
Enantioselective synthesis of spirocyclic aminochroman derivatives according to the CN(R,S) strategy.
|
J Org Chem
|
2003
|
0.75
|
22
|
Synthesis and initial results for MAO-B inhibition by new N-propargyl-3-pyrrol-1-ylindanamine derivatives, analogues of rasagiline.
|
J Enzyme Inhib Med Chem
|
2003
|
0.75
|
23
|
Efficient synthesis and first regioselective C-3 direct arylation of imidazo[1,2-b]pyrazoles.
|
Chemistry
|
2012
|
0.75
|
24
|
New efficient route to dissymmetric 2,4-di(het)aryl-pyrido[3,2-d]pyrimidines via regioselective cross-coupling reactions.
|
Org Lett
|
2007
|
0.75
|
25
|
Tripodal ligand incorporating dual fluorescent ionophore: a coordinative control of photoinduced electron transfer.
|
Photochem Photobiol Sci
|
2003
|
0.75
|
26
|
Efficient metal-free synthesis of various pyrido[2',1':2,3]imidazo- [4,5-b]quinolines.
|
Chemistry
|
2013
|
0.75
|
27
|
Synthesis and evaluation of the antiproliferative activity of novel isoindolo[2,1-a]quinoxaline and indolo[1,2-a]quinoxaline derivatives.
|
J Enzyme Inhib Med Chem
|
2011
|
0.75
|
28
|
Synthesis and in vitro cytostatic activity of new beta-D-arabino furan[1',2':4,5]oxazolo- and arabino-pyrimidinone derivatives.
|
Eur J Med Chem
|
2009
|
0.75
|
29
|
Efficient pallado-catalyzed C6-(het)arylation of Imidazo[1,2-b][1,2,4,5]tetrazines under microwave irradiations.
|
J Comb Chem
|
2010
|
0.75
|
30
|
Anti-leukemia activity of 7-hydroxy-2-substituted-methyl-5H-oxazolo[3,2-a]pyrimidin-5-one derivatives.
|
J Enzyme Inhib Med Chem
|
2002
|
0.75
|
31
|
Potential of immobilized artificial membrane chromatography for lipophilicity determination of arylpropionic acid non-steroidal anti-inflammatory drugs.
|
J Pharm Biomed Anal
|
2003
|
0.75
|
32
|
Synthesis and PC3 androgen-independent prostate cells antiproliferative effect of fagaronine derivatives.
|
J Enzyme Inhib Med Chem
|
2007
|
0.75
|
33
|
Antitumor activity of semisynthetic derivatives of Aconitum alkaloids.
|
Invest New Drugs
|
2013
|
0.75
|
34
|
Derivatization of (+/-)-5-[(2-methylphenoxy)methyl]-2-amino-2-oxazoline, an imidazoline binding sites ligand, with (+)-(R)-alpha-methylbenzyl isocyanate for drug monitoring purposes.
|
J Enzyme Inhib Med Chem
|
2002
|
0.75
|
35
|
Smiles rearrangement as a tool for the preparation of dihydrodipyridopyrazines.
|
Org Lett
|
2009
|
0.75
|