R428, a selective small molecule inhibitor of Axl kinase, blocks tumor spread and prolongs survival in models of metastatic breast cancer.

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🔗 View Article (PMID 20145120)

Published in Cancer Res on February 09, 2010

Authors

Sacha J Holland1, Alison Pan, Christian Franci, Yuanming Hu, Betty Chang, Weiqun Li, Matt Duan, Allan Torneros, Jiaxin Yu, Thilo J Heckrodt, Jing Zhang, Pingyu Ding, Ayodele Apatira, Joanne Chua, Ralf Brandt, Polly Pine, Dane Goff, Rajinder Singh, Donald G Payan, Yasumichi Hitoshi

Author Affiliations

1: Rigel, Inc., 1180 Veteran's Boulevard, South San Francisco, CA 94112, USA. sholland@rigel.com

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