Published in Org Lett on February 21, 2011
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Lead discovery, chemistry optimization, and biological evaluation studies of novel biamide derivatives as CB2 receptor inverse agonists and osteoclast inhibitors. J Med Chem (2012) 0.89
The state of the art of chemical biology. Chembiochem (2009) 0.88
Structure-activity relationship and mechanism of action studies of manzamine analogues for the control of neuroinflammation and cerebral infections. J Med Chem (2010) 0.88
Conformational preferences of natural and C3-modified epothilones in aqueous solution. J Med Chem (2008) 0.88
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Molecular torsion balances: evidence for favorable orthogonal dipolar interactions between organic fluorine and amide groups. Angew Chem Int Ed Engl (2007) 0.87
Total synthesis of (-)-zampanolide and structure-activity relationship studies on (-)-dactylolide derivatives. Chemistry (2012) 0.87
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Stereoselective synthesis of a monocyclic peloruside a analogue. Org Lett (2010) 0.85
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Ginger phenylpropanoids inhibit IL-1beta and prostanoid secretion and disrupt arachidonate-phospholipid remodeling by targeting phospholipases A2. J Immunol (2011) 0.84
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Practical, highly active, and enantioselective ferrocenyl-imidazoline palladacycle catalysts (FIPs) for the aza-Claisen rearrangement of N-para-methoxyphenyl trifluoroacetimidates. Angew Chem Int Ed Engl (2006) 0.83
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Highly potent modulation of GABA(A) receptors by valerenic acid derivatives. ChemMedChem (2010) 0.83
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Perfluorophenyl-phenyl interactions in the crystallization and topochemical polymerization of triacetylene monomers. Chemistry (2009) 0.83
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Molecular recognition at the active site of catechol-O-methyltransferase (COMT): adenine replacements in bisubstrate inhibitors. Chemistry (2011) 0.82
High-affinity inhibitors of tRNA-guanine transglycosylase replacing the function of a structural water cluster. Chemistry (2009) 0.81
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Polymer backbone conformation--a challenging task for database information retrieval. Angew Chem Int Ed Engl (2009) 0.81
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Total synthesis of the marine diterpenoid blumiolide C. Angew Chem Int Ed Engl (2008) 0.80