Discovery of salermide-related sirtuin inhibitors: binding mode studies and antiproliferative effects in cancer cells including cancer stem cells.

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Published in J Med Chem on December 12, 2012

Authors

Dante Rotili1, Domenico Tarantino, Angela Nebbioso, Chantal Paolini, Covadonga Huidobro, Ester Lara, Paolo Mellini, Alessia Lenoci, Riccardo Pezzi, Giorgia Botta, Maija Lahtela-Kakkonen, Antti Poso, Christian Steinkühler, Paola Gallinari, Ruggero De Maria, Mario Fraga, Manel Esteller, Lucia Altucci, Antonello Mai

Author Affiliations

1: Istituto Pasteur-Fondazione Cenci Bolognetti, Dipartimento di Chimica e Tecnologie del Farmaco, Università degli Studi di Roma La Sapienza, P.le A. Moro 5, 00185 Roma, Italy.

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