GABA reduces binding of 3H-methyl beta-carboline-3-carboxylate to brain benzodiazepine receptors.

PubWeight™: 1.00‹?› | Rank: Top 15%

🔗 View Article (PMID 6273744)

Published in Nature on December 03, 1981

Authors

C Braestrup, M Nielsen

Articles by these authors

Confidential inquiry into quality of care before admission to intensive care. BMJ (1998) 11.32

Screening for breast cancer with mammography. Cochrane Database Syst Rev (2006) 5.19

International Union of Pharmacology. XV. Subtypes of gamma-aminobutyric acidA receptors: classification on the basis of subunit structure and receptor function. Pharmacol Rev (1998) 4.37

Specific benzodiazepine receptors in rat brain characterized by high-affinity (3H)diazepam binding. Proc Natl Acad Sci U S A (1977) 3.13

Older persons after hospitalization: a controlled study of home aide service. Am J Public Health (1972) 2.44

Use of a transposon (Tndif) to obtain suppressing and nonsuppressing insertions of the dif resolvase site of Escherichia coli. Genes Dev (1996) 2.42

Differences in risk factors for local and distant recurrence after breast-conserving therapy or mastectomy for stage I and II breast cancer: pooled results of two large European randomized trials. J Clin Oncol (2001) 2.28

Basement membrane changes in breast cancer detected by immunohistochemical staining for laminin. Cancer Res (1981) 2.21

Brain glutamate transporter proteins form homomultimers. J Biol Chem (1996) 2.01

High densities of benzodiazepine receptors in human cortical areas. Nature (1977) 1.97

Somatic APC mosaicism: an underestimated cause of polyposis coli. Gut (2007) 1.79

Evidence for accelerated colorectal adenoma--carcinoma progression in MUTYH-associated polyposis? Gut (2011) 1.74

Interaction of convulsive ligands with benzodiazepine receptors. Science (1982) 1.72

Prediction of protein secondary structure at 80% accuracy. Proteins (2000) 1.65

ABC of intensive care. Criteria for admission. BMJ (1999) 1.65

Task-dependent influences of attention on the activation of human primary visual cortex. Proc Natl Acad Sci U S A (1998) 1.60

SARS CTL vaccine candidates; HLA supertype-, genome-wide scanning and biochemical validation. Tissue Antigens (2004) 1.52

Metastases to the breast from extramammary carcinomas. Acta Pathol Microbiol Scand A (1981) 1.45

Flash pulmonary oedema. Lancet (2001) 1.43

Corpus callosum abnormalities, intellectual disability, speech impairment, and autism in patients with haploinsufficiency of ARID1B. Clin Genet (2011) 1.42

Identification, paracrine generation, and possible function of human breast carcinoma myofibroblasts in culture. In Vitro Cell Dev Biol (1992) 1.41

Constitutive STAT3-activation in Sezary syndrome: tyrphostin AG490 inhibits STAT3-activation, interleukin-2 receptor expression and growth of leukemic Sezary cells. Leukemia (2001) 1.40

Multiplicity in polyp count and extracolonic manifestations in 40 Dutch patients with MYH associated polyposis coli (MAP). J Med Genet (2005) 1.38

Pinocytic activity of rabbit alveolar macrophages in vitro. J Reticuloendothel Soc (1978) 1.28

STAT3-mediated constitutive expression of SOCS-3 in cutaneous T-cell lymphoma. Blood (2001) 1.27

Urinary and brain beta-carboline-3-carboxylates as potent inhibitors of brain benzodiazepine receptors. Proc Natl Acad Sci U S A (1980) 1.25

Inhibition of protein phosphatase 2A induces serine/threonine phosphorylation, subcellular redistribution, and functional inhibition of STAT3. Proc Natl Acad Sci U S A (1999) 1.22

Attention-regulated activity in human primary visual cortex. J Neurophysiol (1998) 1.21

Some properties of brain specific benzodiazepine receptors: new evidence for multiple receptors. Pharmacol Biochem Behav (1979) 1.19

Pharmacological characterization of benzodiazepine receptors in the brain. Eur J Pharmacol (1978) 1.18

Prognosis after treatment for loco-regional recurrence after mastectomy or breast conserving therapy in two randomised trials (EORTC 10801 and DBCG-82TM). EORTC Breast Cancer Cooperative Group and the Danish Breast Cancer Cooperative Group. Eur J Cancer (1999) 1.17

Precancerous and cancerous breast lesions during lifetime and at autopsy. A study of 83 women. Cancer (1984) 1.15

Severe magnesium toxicity after magnesium sulphate enema in a chronically constipated child. BMJ (1990) 1.12

What and when: parallel and convergent processing in motor control. J Neurosci (2000) 1.10

Neural representation of a rhythm depends on its interval ratio. J Neurosci (1999) 1.09

Diazepam-binding inhibitor: a neuropeptide and/or an acyl-CoA ester binding protein? Biochem J (1990) 1.06

Contralateral cancerous breast lesions in women with clinical invasive breast carcinoma. Cancer (1986) 1.04

Complex structure of quisqualate-sensitive glutamate receptors in rat cortex. Neurosci Lett (1985) 1.04

Retinoblastoma among offspring of adult survivors in Denmark. Acta Ophthalmol (Copenh) (1968) 1.04

Biochemical differentiation of amphetamine vs methylphenidate and nomifensine in rats. J Pharm Pharmacol (1977) 1.04

Calcium discriminates two [3H]kainate binding sites with different molecular target sizes in rat cortex. Neurosci Lett (1986) 1.04

In vivo measurement of dopamine receptors in human brain by positron emission tomography. Age and sex differences. Ann N Y Acad Sci (1988) 1.02

Methylphenidate-like effects of the new antidepressant drug nomifensine (HOE 984). Eur J Pharmacol (1976) 1.01

Cutting edge: TCR stimulation by antibody and bacterial superantigen induces Stat3 activation in human T cells. J Immunol (1999) 1.01

Evidence for a late evolutionary appearance of brain-specific benzodiazepine receptors: an investigation of 18 vertebrate and 5 invertebrate species. Brain Res (1978) 1.01

Cystosarcoma phyllodes. A review of 19 cases with emphasis on the occurrence of associated breast carcinoma. Acta Pathol Microbiol Immunol Scand A (1986) 1.01

The role of caspase 3 and BclxL in the action of interleukin 7 (IL-7): a survival factor in activated human T cells. Cytokine (1998) 1.00

[3H]Propyl beta-carboline-3-carboxylate as a selective radioligand for the BZ1 benzodiazepine receptor subclass. J Neurochem (1981) 1.00

Benzodiazepine receptor ligands with positive and negative efficacy. Neuropharmacology (1983) 1.00

Characterization of tiagabine (NO-328), a new potent and selective GABA uptake inhibitor. Eur J Pharmacol (1991) 0.99

The multiligand alpha 2-macroglobulin receptor/low density lipoprotein receptor-related protein (alpha 2MR/LRP). Binding and endocytosis of fluid phase and membrane-associated ligands. Ann N Y Acad Sci (1994) 0.97

Arginine residue 120 of the human GABAA receptor alpha 1, subunit is essential for GABA binding and chloride ion current gating. Neuroreport (1999) 0.95

Histologic changes and silicone concentrations in human breast tissue surrounding silicone breast prostheses. Plast Reconstr Surg (1990) 0.95

Urokinase-type plasminogen activator receptor is internalized by different mechanisms in polarized and nonpolarized Madin-Darby canine kidney epithelial cells. Mol Biol Cell (1999) 0.94

A study of the contribution of hippocampal-accumbens-subpallidal projections to locomotor activity. Behav Neural Biol (1984) 0.93

Brain specific benzodiazepine receptors. Br J Psychiatry (1978) 0.93

Characterization of a kidney proximal tubule cell line, LLC-PK1, expressing endocytotic active megalin. J Am Soc Nephrol (1998) 0.93

Novel plant Ca(2+)-binding protein expressed in response to abscisic acid and osmotic stress. J Biol Chem (1996) 0.92

Differential pharmacological effects of benzodiazepine receptor inverse agonists. Adv Biochem Psychopharmacol (1983) 0.92

High frequency of copy-neutral LOH in MUTYH-associated polyposis carcinomas. J Pathol (2008) 0.92

Suppression of systemic, intramuscular, and subcutaneous adipose tissue lipolysis by insulin in humans. J Clin Endocrinol Metab (2000) 0.91

Ethyl beta-carboline-3-carboxylate shows differential benzodiazepine receptor interaction. Nature (1980) 0.91

Honokiol and magnolol increase the number of [3H] muscimol binding sites three-fold in rat forebrain membranes in vitro using a filtration assay, by allosterically increasing the affinities of low-affinity sites. Neurochem Res (1999) 0.91

Benzodiazepine receptors. Arzneimittelforschung (1980) 0.90

Uptake inhibition of biogenic amines by newer antidepressant drugs: relevance to the dopamine hypothesis of depression. Psychopharmacology (Berl) (1977) 0.90

An autopsy study of radial scar in the female breast. Histopathology (1985) 0.90

Informed choice requires information about both benefits and harms. J Med Ethics (2009) 0.90

Insecticide-treated bed nets reduce plasma antibody levels and limit the repertoire of antibodies to Plasmodium falciparum variant surface antigens. Clin Diagn Lab Immunol (2001) 0.90

Non-NMDA glutamate receptor antagonist 3H-CNOX binds with equal affinity to two agonist states of quisqualate receptors. Biochem Pharmacol (1989) 0.89

Activation of Stat-3 is involved in the induction of apoptosis after ligation of major histocompatibility complex class I molecules on human Jurkat T cells. Blood (1998) 0.89

Hepatic lipase mediates the uptake of chylomicrons and beta-VLDL into cells via the LDL receptor-related protein (LRP). J Lipid Res (1996) 0.89

Classification trees. A possible method for iso-resource grouping in intensive care. Anaesthesia (1998) 0.89

Characterization of the influence of unsaturated free fatty acids on brain GABA/benzodiazepine receptor binding in vitro. J Neurochem (1994) 0.88

FYVE zinc-finger proteins in the plant model Arabidopsis thaliana: identification of PtdIns3P-binding residues by comparison of classic and variant FYVE domains. Biochem J (2001) 0.88

A carboxyl-terminal fragment of lipoprotein lipase binds to the low density lipoprotein receptor-related protein and inhibits lipase-mediated uptake of lipoprotein in cells. J Biol Chem (1994) 0.88

Evaluation of the beta-carboline ZK 93 426 as a benzodiazepine receptor antagonist. Psychopharmacology (Berl) (1984) 0.88

The synthesis of novel GABA uptake inhibitors. 1. Elucidation of the structure-activity studies leading to the choice of (R)-1-[4,4-bis(3-methyl-2-thienyl)-3-butenyl]-3-piperidinecarboxylic acid (tiagabine) as an anticonvulsant drug candidate. J Med Chem (1993) 0.88

On the regulation of sweat secretion in exercise. Acta Physiol Scand (1965) 0.87

Honokiol and magnolol selectively interact with GABAA receptor subtypes in vitro. Pharmacology (2001) 0.87

Interleukin 2 induces a transient downregulation of protein phosphatase 1 and 2A activity in human T cells. Tissue Antigens (1997) 0.87

High affinity of the naturally-occurring biflavonoid, amentoflavon, to brain benzodiazepine receptors in vitro. Biochem Pharmacol (1988) 0.87

The monoamine oxidase B inhibitor deprenyl potentiates phenylethylamine behaviour in rats without inhibition of catecholamine metabolite formation. Eur J Pharmacol (1975) 0.87

Ligands for benzodiazepine receptors with positive and negative efficacy. Biochem Pharmacol (1984) 0.86

Evidence that the anticonflict effect of midazolam in amygdala is mediated by the specific benzodiazepine receptors. Neurosci Lett (1985) 0.86

The apparent target size of rat brain benzodiazepine receptor, acetylcholinesterase, and pyruvate kinase is highly influenced by experimental conditions. J Biol Chem (1988) 0.85

Non-rigid registration by geometry-constrained diffusion. Med Image Anal (2001) 0.85

Inherited predisposition to colorectal adenomas caused by multiple rare alleles of MUTYH but not OGG1, NUDT1, NTH1 or NEIL 1, 2 or 3. Gut (2008) 0.85

Five years experience of breast augmentation using silicone gel prostheses with emphasis on capsule shrinkage. Scand J Plast Reconstr Surg (1984) 0.85

Acquired generalized lipoatrophy (AGL): highly selective MR lipid imaging and localized (1)H-MRS. J Magn Reson Imaging (2000) 0.85

Neuropharmacological evidence to suggest that the nucleus accumbens and subpallidal region contribute to exploratory locomotion. Behav Neural Biol (1984) 0.85

Decreased agonist sensitivity of human GABA(A) receptors by an amino acid variant, isoleucine to valine, in the alpha1 subunit. Eur J Pharmacol (1997) 0.84

Size determination of binding polymers for [3H]imipramine and [3H]paroxetine in human platelet membranes. Eur J Pharmacol (1984) 0.84