Published in Chem Commun (Camb) on September 08, 2005
Novel 2-[(benzylamino)methyl]pyrrolidine-3,4-diol derivatives as alpha-mannosidase inhibitors and with antitumor activities against hematological and solid malignancies. Bioorg Med Chem (2010) 1.40
Rational design of indoleamine 2,3-dioxygenase inhibitors. J Med Chem (2010) 1.22
Organosulfur compounds: electrophilic reagents in transition-metal-catalyzed carbon-carbon bond-forming reactions. Angew Chem Int Ed Engl (2005) 0.99
Recent synthetic approaches toward non-anomeric spiroketals in natural products. Molecules (2008) 0.97
Silyl methallylsulfinates: efficient and powerful agents for the chemoselective silylation of alcohols, polyols, phenols and carboxylic acids. Chem Commun (Camb) (2005) 0.93
Structural insights into the specificity of Xyn10B from Paenibacillus barcinonensis and its improved stability by forced protein evolution. J Biol Chem (2009) 0.91
Synthesis of the C(1)-C(11) polyene fragment of apoptolidin with a new sulfur dioxide-based organic chemistry. Chemistry (2005) 0.90
New efficient route to an advanced precursor of the AB spiroketal of spongistatins. Org Lett (2007) 0.85
Synthesis of novel pyrrolidine 3,4-diol derivatives as inhibitors of alpha-L-fucosidases. Org Biomol Chem (2009) 0.85
Rational design of 4-aryl-1,2,3-triazoles for indoleamine 2,3-dioxygenase 1 inhibition. J Med Chem (2012) 0.85
Scope and limitations of the double [4+3]-cycloadditions of 2-oxyallyl cations to 2,2'-methylenedifuran and derivatives. J Org Chem (2003) 0.84
New synthetic seven-membered 1-azasugars displaying potent inhibition towards glycosidases and glucosylceramide transferase. Chembiochem (2008) 0.84
Short synthesis of the C16-C28 polyketide fragment of apoptolidin A aglycone. Chem Commun (Camb) (2007) 0.83
Palladium-catalyzed Stille cross-couplings of sulfonyl chlorides and organostannanes. J Am Chem Soc (2003) 0.82
Total synthesis and determination of the absolute configuration of (-)-dolabriferol. Angew Chem Int Ed Engl (2010) 0.82
New concise total synthesis of (+)-lentiginosine and some structural analogues. J Org Chem (2005) 0.81
Synthesis and conformational analysis of (alpha-D-galactosyl)phenylmethane and alpha-,beta-difluoromethane analogues: interactions with the plant lectin viscumin. Chemistry (2009) 0.81
Synthesis and anti-HIV activity of trivalent CD4-mimetic miniproteins. Bioorg Med Chem (2007) 0.80
Functionalized pyrrolidines inhibit alpha-mannosidase activity and growth of human glioblastoma and melanoma cells. J Med Chem (2005) 0.80
Glycosidase inhibitors as potential HIV entry inhibitors? Curr Drug Metab (2004) 0.79
Palladium-catalyzed Suzuki-Miyaura cross-couplings of sulfonyl chlorides and boronic acids. Org Lett (2004) 0.79
Search for alpha-glucosidase inhibitors: new N-substituted valienamine and conduramine F-1 derivatives. Bioorg Med Chem (2006) 0.79
Tandem Staudinger-azaWittig mediated ring expansion: rapid access to new isofagomine-tetrahydroxyazepane hybrids. Chem Commun (Camb) (2006) 0.79
Iron-catalyzed desulfinylative C-C cross-coupling reactions of sulfonyl chlorides with grignard reagents. Angew Chem Int Ed Engl (2008) 0.79
An efficient combinatorial method for the discovery of glycosidase inhibitors. Chembiochem (2002) 0.78
Stereoselective syntheses of 1,4-dideoxy-1,4-imino-octitols and novel tetrahydroxyindolizidines. J Org Chem (2003) 0.78
Chemoselective C-H bond activation: ligand and solvent free iron-catalyzed oxidative C-C cross-coupling of tertiary amines with terminal alkynes. Reaction scope and mechanism. Org Lett (2009) 0.78
A C-linked disaccharide analogue of Thomsen-Friedenreich epitope induces a strong immune response in mice. Chemistry (2012) 0.78
6-Azido hyacinthacine A2 gives a straightforward access to the first multivalent pyrrolizidine architectures. Org Biomol Chem (2014) 0.78
Nucleophilic opening of epoxyazepanes: expanding the family of polyhydroxyazepane-based glycosidase inhibitors. Org Biomol Chem (2006) 0.78
Design and synthesis of acetamido tri- and tetra-hydroxyazepanes: potent and selective beta-N-acetylhexosaminidase inhibitors. Bioorg Med Chem (2009) 0.78
Total asymmetric synthesis of (-)-conduramine B-1 and of its enantiomer. N-Benzyl derivatives of conduramine B-1 are beta-glucosidase inhibitors. Bioorg Med Chem Lett (2005) 0.78
Desulfinylation of prop-2-enesulfinic acid: experimental results and mechanistic theoretical analysis. J Am Chem Soc (2009) 0.77
Sulfur dioxide mediated one-pot, three- and four-component syntheses of polyfunctional sulfonamides and sulfonic esters: study of the stereoselectivity of the ene reaction of sulfur dioxide. J Org Chem (2004) 0.77
Synthesis of optically active 5-alkoxy-6-methylcyclohex-2-en-1-ones and 4-alkoxy-5-methylcyclopent-1-enyl benzoate. J Org Chem (2009) 0.77
Synthesis of new oxathiazinane dioxides and their in vitro cancer cell growth inhibitory activity. Bioorg Med Chem Lett (2009) 0.77
The first synthesis of substituted azepanes mimicking monosaccharides: a new class of potent glycosidase inhibitors. Org Biomol Chem (2004) 0.77
Synthesis of (E,Z)-1-alkoxy-3-acyloxy-2-methylpenta-1,3-dienes via Danishefsky-type dienes or O-acylation of enones. J Org Chem (2009) 0.77
Ab initio and experimental studies on the hetero-Diels-Alder and cheletropic additions of sulfur dioxide to (E)-1-methoxybutadiene: a mechanism involving three molecules of SO(2). J Org Chem (2002) 0.77
Concise synthesis of complicated polypropionates through one-pot dissymmetrical two-directional chain elongation. Chemistry (2011) 0.76
Polysulfones: catalysts for alkene isomerization. Angew Chem Int Ed Engl (2004) 0.76
Three dimensional structure of a bacterial α-l-fucosidase with a 5-membered iminocyclitol inhibitor. Bioorg Med Chem (2013) 0.76
Anti-cancer activity of 5-O-alkyl 1,4-imino-1,4-dideoxyribitols. Bioorg Med Chem (2011) 0.76
The anti-lymphoma activity of APO866, an inhibitor of nicotinamide adenine dinucleotide biosynthesis, is potentialized when used in combination with anti-CD20 antibody. Leuk Lymphoma (2014) 0.76
Amine-linked diglycosides: Synthesis facilitated by the enhanced reactivity of allylic electrophiles, and glycosidase inhibition assays. Beilstein J Org Chem (2011) 0.76
Effects of ethylene glycol addition on the aggregation and micellar growth of gemini surfactants. Langmuir (2006) 0.76
Specific activation of ERK pathways by chitin oligosaccharides in embryonic zebrafish cell lines. Glycobiology (2003) 0.76
Total asymmetric syntheses of β-hydroxy-δ-lactones via Umpolung with sulfur dioxide. J Org Chem (2011) 0.75
Palladium-catalyzed conversion of beta,gamma-unsaturated silyl sulfinates into (E)-alkenes: asymmetric synthesis of polypropionate fragments. J Org Chem (2004) 0.75
Synthesis of long-chain polyketide fragments by reaction of 1,3-dioxy-1,3-dienes with allylsilanes: umpolung with sulfur dioxide. Org Lett (2004) 0.75
Syntheses and biological activities of 1,4-iminoalditol derivatives as alpha-L-fucosidase inhibitors. Chimia (Aarau) (2011) 0.75
Allyl, methallyl, prenyl, and methylprenyl ethers as protected alcohols: their selective cleavage with diphenyldisulfone under neutral conditions. Org Lett (2004) 0.75
Synthesis of branched seven-membered 1-N-iminosugars and their evaluation as glycosidase inhibitors. Carbohydr Res (2011) 0.75
Synthesis and glycosidase inhibitory activities of 2-(aminoalkyl)pyrrolidine-3,4-diol derivatives. Bioorg Med Chem (2003) 0.75
Hetaryleneaminopolyols and hetarylenecarbopeptoids: a new type of glyco- and peptidomimetics. Syntheses and studies on solution conformation and dynamics. J Org Chem (2003) 0.75
Amide formation in one pot from carboxylic acids and amines via carboxyl and sulfinyl mixed anhydrides. Org Lett (2013) 0.75
Synthesis of enantiomerically pure 1,2-diamine derivatives of 7-azabicyclo[2.2.1]heptane. New leads as glycosidase inhibitors and rigid scaffolds for the preparation of peptide analogues. J Org Chem (2003) 0.75
Mechanism of the diphenyldisulfone-catalyzed isomerization of alkenes. Origin of the chemoselectivity: experimental and quantum chemistry studies. J Am Chem Soc (2006) 0.75
First asymmetric synthesis of the cyclohexanone subunit of baconipyrones A and B. Revision of its structure. Org Lett (2004) 0.75
Synthesis of d- and l-2,3-trans-3,4-cis-4,5-trans-3,4-dihydroxy-5-hydroxymethylproline and tripeptides containing them. J Org Chem (2004) 0.75
Monosaccharides and analogues from simple achiral unsaturated compounds. Chimia (Aarau) (2011) 0.75
Amides in one pot from carboxylic acids and amines via sulfinylamides. Org Lett (2014) 0.75
The hetero-Diels-Alder addition of sulfur dioxide: the pseudo-chair conformation of a 4,5-dialkylsultine. Chemistry (2003) 0.75
A short and convenient synthesis of 1-deoxymannojirimycin and N-oxy analogues from D-fructose. J Org Chem (2009) 0.75
Total asymmetric synthesis of monosaccharides and analogues. Chimia (Aarau) (2011) 0.75
Synthesis of [(2S,3S,4R)-3,4-dihydroxypyrrolidin-2-yl]-5-methylfuran-4-carboxylic acid derivatives: new leads as selective beta-galactosidase inhibitors. Bioorg Med Chem Lett (2002) 0.75
Synthesis and conformational analysis of novel trimeric maleimide cross-linking reagents. J Org Chem (2007) 0.75
Short diastereoselective synthesis of the C1-C13 (AB spiroacetal) and C17-C28 fragments (CD spiroacetal) of spongistatin 1 and 2 through double chain-elongation reactions. Chemistry (2010) 0.75
Equilibrium and kinetic deuterium isotope effects on the hetero-Diels-Alder addition of sulfur dioxide. Angew Chem Int Ed Engl (2003) 0.75
Physicochemical characterization of bromide mono- and dimeric surfactants with phenyl and cyclohexyl rings in the head group. J Colloid Interface Sci (2011) 0.75
The norbornene mystery revealed. Chem Commun (Camb) (2010) 0.75
Exploiting the ring strain in bicyclo[2.2.1]heptane systems for the stereoselective preparation of highly functionalized cyclopentene, dihydrofuran, pyrroline, and pyrrolidine scaffolds. Org Lett (2011) 0.75
Rapid discovery of potent α-fucosidase inhibitors by in situ screening of a library of (pyrrolidin-2-yl)triazoles. Org Biomol Chem (2014) 0.75
Synthesis and inhibitory activities of novel C-3 substituted azafagomines: a new type of selective inhibitors of α-L-fucosidases. Bioorg Med Chem (2010) 0.75
Strain-promoted retro-Dieckmann-type condensation on [2.2.2]- and [2.2.1]bicyclic systems: a fragmentation reaction for the preparation of functionalized heterocycles and carbocycles. Org Biomol Chem (2013) 0.75
Glycochemistry today. Chimia (Aarau) (2011) 0.75
Synthesis, biological evaluation, WAC and NMR studies of S-galactosides and non-carbohydrate ligands of cholera toxin based on polyhydroxyalkylfuroate moieties. Chemistry (2013) 0.75
Carbohydrates in sustainable development, Part 1. Renewable resources for chemistry and biotechnology. Preface. Top Curr Chem (2010) 0.75
Allenyl sulfones and allenyl sulfides in the synthesis of 3-pyrrolines. A novel nucleophilic [3 + 2] cycloaddition on allenyl sulfones giving rearranged cycloadducts. Org Lett (2009) 0.75
Synthesis and physicochemical characterization of alkanedyil-α-ω-bis(dimethyldodecylammonium) bromide, 12-s-12,2Br-, surfactants with s=7, 9, 11 in aqueous medium. J Colloid Interface Sci (2012) 0.75