Published in Org Lett on December 03, 2009
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Synthesis and anti-leishmanial activity of heterocyclic betulin derivatives. Bioorg Med Chem (2010) 0.87
Inhibitory effect of the natural product betulin and its derivatives against the intracellular bacterium Chlamydia pneumoniae. Biochem Pharmacol (2010) 0.85
Stereochemical sensitivity of the human UDP-glucuronosyltransferases 2B7 and 2B17. J Med Chem (2006) 0.85
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Design, synthesis, and biological activity of isophthalic acid derivatives targeted to the C1 domain of protein kinase C. J Med Chem (2009) 0.81
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A new insight into solid-state conformation of macrolide antibiotics. Bioorg Med Chem (2007) 0.80
HIV-1 Tat-peptide inhibits protein kinase C and protein kinase A through substrate competition. Eur J Pharm Sci (2010) 0.80
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Synthesis and evaluation of library of betulin derivatives against the botulinum neurotoxin A protease. Bioorg Med Chem Lett (2011) 0.78
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Chiral distinction between the enantiomers of bicyclic alcohols by UDP-glucuronosyltransferases 2B7 and 2B17. Biol Chem (2006) 0.78
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Isoform-selective inhibition of the human UDP-glucuronosyltransferase 2B7 by isolongifolol derivatives. J Med Chem (2007) 0.77
Conformation study of 2-arylbenzimidazoles as inhibitors of Chlamydia pneumoniae growth. Bioorg Med Chem Lett (2012) 0.76
Glucuronidation of psilocin and 4-hydroxyindole by the human UDP-glucuronosyltransferases. Drug Metab Dispos (2009) 0.76
The C1 domain-targeted isophthalate derivative HMI-1b11 promotes neurite outgrowth and GAP-43 expression through PKCα activation in SH-SY5Y cells. Pharmacol Res (2013) 0.76
Exploring the scope of the 29G12 antibody catalyzed 1,3-dipolar cycloaddition reaction. J Org Chem (2005) 0.75
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Synthesis and characterization of hydroxylated mesocarb metabolites for doping control. Arch Pharm (Weinheim) (2009) 0.75
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Stereochemical and steric control of the UDP-glucuronosyltransferase-catalyzed conjugation reaction: a rational approach for the design of inhibitors for the human UGT2B7. ChemMedChem (2007) 0.75
Toxicity of betulin derivatives and in vitro effect on promastigotes and amastigotes of Leishmania infantum and L. donovani. J Antibiot (Tokyo) (2011) 0.75
Synthesis, structure characterization, and enzyme screening of clenbuterol glucuronides. Eur J Pharm Sci (2009) 0.75
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Potent inhibitors of the human UDP-glucuronosyltransferase 2B7 derived from the sesquiterpenoid alcohol longifolol. ChemMedChem (2007) 0.75
Mechanism of the Oxidation of Heptafulvenes to Tropones Studied by Online Mass Spectrometry and Density Functional Theory Calculations. J Org Chem (2019) 0.75
A modification of the Hammett equation for predicting ionisation constants of p-vinyl phenols. Eur J Pharm Sci (2005) 0.75
Microplate screening assay for binding of ligands to bovine or reindeer beta-lactoglobulins. J Biochem Biophys Methods (2006) 0.75
Structural Isosteres of Phosphate Groups in the Protein Data Bank. J Chem Inf Model (2017) 0.75
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Electrospray ionization mass spectrometry and tandem mass spectrometry of clodronate and related bisphosphonate and phosphonate compounds. J Mass Spectrom (2002) 0.75
On the hydrolytic behavior of tinidazole, metronidazole, and ornidazole. J Pharm Sci (2003) 0.75