PubRank

Pierre Vogel

Author PubWeight™ 36.58‹?›

Top papers

Rank Title Journal Year PubWeight™‹?›
1 Novel 2-[(benzylamino)methyl]pyrrolidine-3,4-diol derivatives as alpha-mannosidase inhibitors and with antitumor activities against hematological and solid malignancies. Bioorg Med Chem 2010 1.40
2 Rational design of indoleamine 2,3-dioxygenase inhibitors. J Med Chem 2010 1.22
3 Organosulfur compounds: electrophilic reagents in transition-metal-catalyzed carbon-carbon bond-forming reactions. Angew Chem Int Ed Engl 2005 0.99
4 Recent synthetic approaches toward non-anomeric spiroketals in natural products. Molecules 2008 0.97
5 Silyl methallylsulfinates: efficient and powerful agents for the chemoselective silylation of alcohols, polyols, phenols and carboxylic acids. Chem Commun (Camb) 2005 0.93
6 Structural insights into the specificity of Xyn10B from Paenibacillus barcinonensis and its improved stability by forced protein evolution. J Biol Chem 2009 0.91
7 Synthesis of the C(1)-C(11) polyene fragment of apoptolidin with a new sulfur dioxide-based organic chemistry. Chemistry 2005 0.90
8 Rational design of 4-aryl-1,2,3-triazoles for indoleamine 2,3-dioxygenase 1 inhibition. J Med Chem 2012 0.85
9 Synthesis of novel pyrrolidine 3,4-diol derivatives as inhibitors of alpha-L-fucosidases. Org Biomol Chem 2009 0.85
10 New efficient route to an advanced precursor of the AB spiroketal of spongistatins. Org Lett 2007 0.85
11 Scope and limitations of the double [4+3]-cycloadditions of 2-oxyallyl cations to 2,2'-methylenedifuran and derivatives. J Org Chem 2003 0.84
12 New synthetic seven-membered 1-azasugars displaying potent inhibition towards glycosidases and glucosylceramide transferase. Chembiochem 2008 0.84
13 Short synthesis of the C16-C28 polyketide fragment of apoptolidin A aglycone. Chem Commun (Camb) 2007 0.83
14 Total synthesis and determination of the absolute configuration of (-)-dolabriferol. Angew Chem Int Ed Engl 2010 0.82
15 Palladium-catalyzed Stille cross-couplings of sulfonyl chlorides and organostannanes. J Am Chem Soc 2003 0.82
16 New concise total synthesis of (+)-lentiginosine and some structural analogues. J Org Chem 2005 0.81
17 Synthesis and conformational analysis of (alpha-D-galactosyl)phenylmethane and alpha-,beta-difluoromethane analogues: interactions with the plant lectin viscumin. Chemistry 2009 0.81
18 Functionalized pyrrolidines inhibit alpha-mannosidase activity and growth of human glioblastoma and melanoma cells. J Med Chem 2005 0.80
19 Tandem Staudinger-azaWittig mediated ring expansion: rapid access to new isofagomine-tetrahydroxyazepane hybrids. Chem Commun (Camb) 2006 0.79
20 Glycosidase inhibitors as potential HIV entry inhibitors? Curr Drug Metab 2004 0.79
21 Search for alpha-glucosidase inhibitors: new N-substituted valienamine and conduramine F-1 derivatives. Bioorg Med Chem 2006 0.79
22 Palladium-catalyzed Suzuki-Miyaura cross-couplings of sulfonyl chlorides and boronic acids. Org Lett 2004 0.79
23 The hetero-Diels-Alder addition of sulfur dioxide to 1-fluorobuta-1,3-dienes: the sofa conformations preferred by 6-fluorosultines (6-fluoro-3,6-dihydro-1,2-oxathiin-2-oxides) enjoy enthalpic and conformational Anomeric effects. Chemistry 2002 0.79
24 Iron-catalyzed desulfinylative C-C cross-coupling reactions of sulfonyl chlorides with grignard reagents. Angew Chem Int Ed Engl 2008 0.79
25 A C-linked disaccharide analogue of Thomsen-Friedenreich epitope induces a strong immune response in mice. Chemistry 2012 0.78
26 Nucleophilic opening of epoxyazepanes: expanding the family of polyhydroxyazepane-based glycosidase inhibitors. Org Biomol Chem 2006 0.78
27 Design and synthesis of acetamido tri- and tetra-hydroxyazepanes: potent and selective beta-N-acetylhexosaminidase inhibitors. Bioorg Med Chem 2009 0.78
28 Total asymmetric synthesis of (-)-conduramine B-1 and of its enantiomer. N-Benzyl derivatives of conduramine B-1 are beta-glucosidase inhibitors. Bioorg Med Chem Lett 2005 0.78
29 An efficient combinatorial method for the discovery of glycosidase inhibitors. Chembiochem 2002 0.78
30 Chemoselective C-H bond activation: ligand and solvent free iron-catalyzed oxidative C-C cross-coupling of tertiary amines with terminal alkynes. Reaction scope and mechanism. Org Lett 2009 0.78
31 Stereoselective syntheses of 1,4-dideoxy-1,4-imino-octitols and novel tetrahydroxyindolizidines. J Org Chem 2003 0.78
32 Synthesis of optically active 5-alkoxy-6-methylcyclohex-2-en-1-ones and 4-alkoxy-5-methylcyclopent-1-enyl benzoate. J Org Chem 2009 0.77
33 Ab initio and experimental studies on the hetero-Diels-Alder and cheletropic additions of sulfur dioxide to (E)-1-methoxybutadiene: a mechanism involving three molecules of SO(2). J Org Chem 2002 0.77
34 Synthesis of new oxathiazinane dioxides and their in vitro cancer cell growth inhibitory activity. Bioorg Med Chem Lett 2009 0.77
35 Desulfinylation of prop-2-enesulfinic acid: experimental results and mechanistic theoretical analysis. J Am Chem Soc 2009 0.77
36 The first synthesis of substituted azepanes mimicking monosaccharides: a new class of potent glycosidase inhibitors. Org Biomol Chem 2004 0.77
37 Sulfur dioxide mediated one-pot, three- and four-component syntheses of polyfunctional sulfonamides and sulfonic esters: study of the stereoselectivity of the ene reaction of sulfur dioxide. J Org Chem 2004 0.77
38 Synthesis of (E,Z)-1-alkoxy-3-acyloxy-2-methylpenta-1,3-dienes via Danishefsky-type dienes or O-acylation of enones. J Org Chem 2009 0.77
39 Concise synthesis of complicated polypropionates through one-pot dissymmetrical two-directional chain elongation. Chemistry 2011 0.76
40 The anti-lymphoma activity of APO866, an inhibitor of nicotinamide adenine dinucleotide biosynthesis, is potentialized when used in combination with anti-CD20 antibody. Leuk Lymphoma 2014 0.76
41 Anti-cancer activity of 5-O-alkyl 1,4-imino-1,4-dideoxyribitols. Bioorg Med Chem 2011 0.76
42 Polysulfones: catalysts for alkene isomerization. Angew Chem Int Ed Engl 2004 0.76
43 Palladium-catalyzed desulfitative Mizoroki-Heck couplings of sulfonyl chlorides with mono- and disubstituted olefins: rhodium-catalyzed desulfitative heck-type reactions under phosphine- and base-free conditions. Chemistry 2005 0.76
44 Total asymmetric syntheses of β-hydroxy-δ-lactones via Umpolung with sulfur dioxide. J Org Chem 2011 0.75
45 Expeditious asymmetric synthesis of a stereoheptad corresponding to the C(19)-C(27)-ansa chain of rifamycins: formal total synthesis of Rifamycin S. Chemistry 2005 0.75
46 Polysulfones: solid organic catalysts for the chemoselective cleavage of methyl-substituted allyl ethers under neutral conditions. Chem Commun (Camb) 2004 0.75
47 Synthesis of branched seven-membered 1-N-iminosugars and their evaluation as glycosidase inhibitors. Carbohydr Res 2011 0.75
48 Spirocyclopropyl pyrrolidines as a new series of alpha-L-fucosidase inhibitors. Bioorg Med Chem 2006 0.75
49 Synthesis of enantiomerically pure 1,2-diamine derivatives of 7-azabicyclo[2.2.1]heptane. New leads as glycosidase inhibitors and rigid scaffolds for the preparation of peptide analogues. J Org Chem 2003 0.75
50 The hetero-Diels-Alder addition of sulfur dioxide: the pseudo-chair conformation of a 4,5-dialkylsultine. Chemistry 2003 0.75
51 Mechanism of the diphenyldisulfone-catalyzed isomerization of alkenes. Origin of the chemoselectivity: experimental and quantum chemistry studies. J Am Chem Soc 2006 0.75
52 The spirocyclopropyl moiety as a methyl surrogate in the structure of l-fucosidase and l-rhamnosidase inhibitors. Bioorg Med Chem 2009 0.75
53 The use of levoglucosenone and isolevoglucosenone as templates for the construction of C-linked disaccharides. Carbohydr Res 2006 0.75
54 The catalyzed desulfinylative allylation of carbonyl compounds with alk-2-enesulfonyl chlorides and silyl alk-2-enesulfinates. Chemistry 2010 0.75
55 Glycochemistry today. Chimia (Aarau) 2011 0.75
56 BCl3-mediated ene reaction of sulfur dioxide and unfunctionalized alkenes. Chemistry 2010 0.75
57 A short and convenient synthesis of 1-deoxymannojirimycin and N-oxy analogues from D-fructose. J Org Chem 2009 0.75
58 Allyl, methallyl, prenyl, and methylprenyl ethers as protected alcohols: their selective cleavage with diphenyldisulfone under neutral conditions. Org Lett 2004 0.75
59 Amide formation in one pot from carboxylic acids and amines via carboxyl and sulfinyl mixed anhydrides. Org Lett 2013 0.75
60 Stereoselective synthesis of (2S,3S,4R,5S)-5-methylpyrrolidine-3,4-diol derivatives that are highly selective alpha-L-fucosidase inhibitors. Chem Commun (Camb) 2005 0.75
61 The norbornene mystery revealed. Chem Commun (Camb) 2010 0.75
62 Synthesis of long-chain polyketide fragments by reaction of 1,3-dioxy-1,3-dienes with allylsilanes: umpolung with sulfur dioxide. Org Lett 2004 0.75
63 Synthesis of d- and l-2,3-trans-3,4-cis-4,5-trans-3,4-dihydroxy-5-hydroxymethylproline and tripeptides containing them. J Org Chem 2004 0.75
64 Synthesis and glycosidase inhibitory activities of 2-(aminoalkyl)pyrrolidine-3,4-diol derivatives. Bioorg Med Chem 2003 0.75
65 First asymmetric synthesis of the cyclohexanone subunit of baconipyrones A and B. Revision of its structure. Org Lett 2004 0.75
66 Palladium-catalyzed conversion of beta,gamma-unsaturated silyl sulfinates into (E)-alkenes: asymmetric synthesis of polypropionate fragments. J Org Chem 2004 0.75
67 Carbohydrates in sustainable development, Part 1. Renewable resources for chemistry and biotechnology. Preface. Top Curr Chem 2010 0.75
68 C-linked disaccharide analogue of the Thomsen-Friedenreich (T)-epitope alpha-O-conjugated to L-serine. Chemistry 2005 0.75
69 Short diastereoselective synthesis of the C1-C13 (AB spiroacetal) and C17-C28 fragments (CD spiroacetal) of spongistatin 1 and 2 through double chain-elongation reactions. Chemistry 2010 0.75
70 Synthesis and glycosidase inhibitory activity of 1-amino-3,6-anhydro-1-deoxy-D-sorbitol derivatives. Bioorg Chem 2009 0.75
71 Synthesis of [(2S,3S,4R)-3,4-dihydroxypyrrolidin-2-yl]-5-methylfuran-4-carboxylic acid derivatives: new leads as selective beta-galactosidase inhibitors. Bioorg Med Chem Lett 2002 0.75
72 Equilibrium and kinetic deuterium isotope effects on the hetero-Diels-Alder addition of sulfur dioxide. Angew Chem Int Ed Engl 2003 0.75
73 Sulfur dioxide-mediated syntheses of polyfunctional alkenes and (E,Z)- and (E,E)-2,4-dien-1-ones. Org Lett 2005 0.75
74 Amides in one pot from carboxylic acids and amines via sulfinylamides. Org Lett 2014 0.75