PubRank

Valery V Fokin

Author PubWeight™ 123.14‹?›

Top papers

Rank Title Journal Year PubWeight™‹?›
1 A stepwise huisgen cycloaddition process: copper(I)-catalyzed regioselective "ligation" of azides and terminal alkynes. Angew Chem Int Ed Engl 2002 24.12
2 Polytriazoles as copper(I)-stabilizing ligands in catalysis. Org Lett 2004 5.49
3 Bioconjugation by copper(I)-catalyzed azide-alkyne [3 + 2] cycloaddition. J Am Chem Soc 2003 5.34
4 Copper(I)-catalyzed synthesis of azoles. DFT study predicts unprecedented reactivity and intermediates. J Am Chem Soc 2005 2.75
5 Copper-catalyzed azide-alkyne cycloaddition (CuAAC) and beyond: new reactivity of copper(I) acetylides. Chem Soc Rev 2010 2.68
6 Mechanism of the ligand-free CuI-catalyzed azide-alkyne cycloaddition reaction. Angew Chem Int Ed Engl 2005 2.62
7 Ruthenium-catalyzed cycloaddition of alkynes and organic azides. J Am Chem Soc 2005 2.35
8 "On water": unique reactivity of organic compounds in aqueous suspension. Angew Chem Int Ed Engl 2005 2.21
9 Efficiency and fidelity in a click-chemistry route to triazole dendrimers by the copper(i)-catalyzed ligation of azides and alkynes. Angew Chem Int Ed Engl 2004 2.11
10 Copper(I)-catalyzed cycloaddition of organic azides and 1-iodoalkynes. Angew Chem Int Ed Engl 2009 2.10
11 Discovery and characterization of catalysts for azide-alkyne cycloaddition by fluorescence quenching. J Am Chem Soc 2004 1.89
12 Rhodium-catalyzed transannulation of 1,2,3-triazoles with nitriles. J Am Chem Soc 2008 1.86
13 Rhodium-catalyzed enantioselective cyclopropanation of olefins with N-sulfonyl 1,2,3-triazoles. J Am Chem Soc 2009 1.85
14 Ruthenium-catalyzed azide-alkyne cycloaddition: scope and mechanism. J Am Chem Soc 2008 1.76
15 Ligand-accelerated Cu-catalyzed azide-alkyne cycloaddition: a mechanistic report. J Am Chem Soc 2007 1.72
16 Iterative in situ click chemistry creates antibody-like protein-capture agents. Angew Chem Int Ed Engl 2009 1.64
17 Inhibitors of HIV-1 protease by using in situ click chemistry. Angew Chem Int Ed Engl 2006 1.63
18 A potent and highly selective inhibitor of human alpha-1,3-fucosyltransferase via click chemistry. J Am Chem Soc 2003 1.53
19 Synthesis and reactivity of rhodium(II) N-triflyl azavinyl carbenes. J Am Chem Soc 2010 1.45
20 Organic synthesis "on water". Chem Rev 2009 1.37
21 Multivalent, bifunctional dendrimers prepared by click chemistry. Chem Commun (Camb) 2005 1.32
22 The allylic azide rearrangement: achieving selectivity. J Am Chem Soc 2005 1.30
23 Practical synthesis of amides from in situ generated copper(I) acetylides and sulfonyl azides. Angew Chem Int Ed Engl 2006 1.29
24 Click chemistry: function follows form. Chem Soc Rev 2010 1.23
25 Catalytic asymmetric C-H insertions of rhodium(II) azavinyl carbenes. J Am Chem Soc 2011 1.22
26 Efficient synthesis of 1-sulfonyl-1,2,3-triazoles. Org Lett 2010 1.19
27 Refinement of structural leads for centrally acting oxime reactivators of phosphylated cholinesterases. J Biol Chem 2012 1.18
28 Ruthenium-catalyzed cycloaddition of aryl azides and alkynes. Org Lett 2007 1.16
29 Efficient synthesis of 2-substituted-1,2,3-triazoles. Org Lett 2008 1.15
30 One-pot synthesis of 1,4-disubstituted 1,2,3-triazoles from in situ generated azides. Org Lett 2004 1.14
31 Copper-catalyzed synthesis of N-sulfonyl-1,2,3-triazoles: controlling selectivity. Angew Chem Int Ed Engl 2007 1.14
32 New structural scaffolds for centrally acting oxime reactivators of phosphylated cholinesterases. J Biol Chem 2011 1.14
33 Rapid diversity-oriented synthesis in microtiter plates for in situ screening of HIV protease inhibitors. Chembiochem 2003 1.13
34 Direct synthesis of 1,5-disubstituted-4-magnesio-1,2,3-triazoles, revisited. Org Lett 2004 1.13
35 One-pot copper(I)-catalyzed synthesis of 3,5-disubstituted isoxazoles. J Org Chem 2005 1.13
36 A microwave-assisted click chemistry synthesis of 1,4-disubstituted 1,2,3-triazoles via a copper(I)-catalyzed three-component reaction. Org Lett 2004 1.13
37 Copper-catalyzed reaction cascade: direct conversion of alkynes into N-sulfonylazetidin-2-imines. Angew Chem Int Ed Engl 2006 1.08
38 Inhibitors of VIM-2 by screening pharmacologically active and click-chemistry compound libraries. Bioorg Med Chem 2009 1.02
39 Oxime-assisted acetylcholinesterase catalytic scavengers of organophosphates that resist aging. J Biol Chem 2011 1.01
40 Arylation of rhodium(II) azavinyl carbenes with boronic acids. J Am Chem Soc 2012 0.99
41 Generation of candidate ligands for nicotinic acetylcholine receptors via in situ click chemistry with a soluble acetylcholine binding protein template. J Am Chem Soc 2012 0.99
42 Rapid discovery and structure-activity profiling of novel inhibitors of human immunodeficiency virus type 1 protease enabled by the copper(I)-catalyzed synthesis of 1,2,3-triazoles and their further functionalization. J Med Chem 2006 0.98
43 Mechanistic studies on the Cu-catalyzed three-component reactions of sulfonyl azides, 1-alkynes and amines, alcohols, or water: dichotomy via a common pathway. J Org Chem 2008 0.98
44 Synthesis and electrochemistry of 2-ethenyl and 2-ethanyl derivatives of 5-nitroimidazole and antimicrobial activity against Giardia lamblia. J Med Chem 2009 0.97
45 Identification of a new endogenous metabolite and the characterization of its protein interactions through an immobilization approach. J Am Chem Soc 2009 0.96
46 Transition-metal-free catalytic synthesis of 1,5-diaryl-1,2,3-triazoles. Org Lett 2010 0.96
47 Design, synthesis and bioactions of novel stable mimetics of lipoxins and aspirin-triggered lipoxins. Prostaglandins Leukot Essent Fatty Acids 2005 0.95
48 Click and pick: identification of sialoside analogues for siglec-based cell targeting. Angew Chem Int Ed Engl 2012 0.92
49 Reactivity of N-(1,2,4-triazolyl)-substituted 1,2,3-triazoles. Org Lett 2011 0.91
50 Sulfonyl-1,2,3-triazoles: convenient synthones for heterocyclic compounds. Angew Chem Int Ed Engl 2012 0.90
51 Ring expansion and rearrangements of rhodium(II) azavinyl carbenes. Angew Chem Int Ed Engl 2012 0.89
52 Expanded therapeutic potential in activity space of next-generation 5-nitroimidazole antimicrobials with broad structural diversity. Proc Natl Acad Sci U S A 2013 0.89
53 Rhodium(II)-catalyzed asymmetric sulfur(VI) reduction of diazo sulfonylamidines. J Am Chem Soc 2012 0.88
54 REGIOSELECTIVE SYNTHESIS OF EITHER 1H- OR 2H-1,2,3- TRIAZOLES VIA MICHAEL ADDITION TO α,ß-UNSATURATED KETONES. Heterocycles 2008 0.87
55 Transannulation of 1-sulfonyl-1,2,3-triazoles with heterocumulenes. J Am Chem Soc 2013 0.87
56 Efficient synthesis of sulfonyl azides from sulfonamides. Org Lett 2008 0.87
57 Antiviral stilbene 1,2-diamines prevent initiation of hepatitis C virus RNA replication at the outset of infection. J Virol 2011 0.86
58 Ultrasound-promoted copper-catalyzed azide-alkyne cycloaddition. J Comb Chem 2010 0.85
59 Imidazole aldoximes effective in assisting butyrylcholinesterase catalysis of organophosphate detoxification. J Med Chem 2014 0.84
60 Stereoselective 1,3-insertions of rhodium(II) azavinyl carbenes. J Am Chem Soc 2013 0.82
61 Centrally acting oximes in reactivation of tabun-phosphoramidated AChE. Chem Biol Interact 2012 0.82
62 Ruthenium-catalyzed cycloaddition of nitrile oxides and alkynes: practical synthesis of isoxazoles. Angew Chem Int Ed Engl 2008 0.81
63 Synthesis and reactivity of sulfamoyl azides and 1-sulfamoyl-1,2,3-triazoles. Org Lett 2011 0.81
64 NH-1,2,3-Triazole-based Inhibitors of the VIM-2 Metallo-β-Lactamase: Synthesis and Structure-Activity Studies. ACS Med Chem Lett 2010 0.81
65 Synthesis of selective agonists for the α7 nicotinic acetylcholine receptor with in situ click-chemistry on acetylcholine-binding protein templates. Mol Pharmacol 2012 0.80
66 Copper(I)-catalyzed cycloaddition of bismuth(III) acetylides with organic azides: synthesis of stable triazole anion equivalents. Angew Chem Int Ed Engl 2013 0.79
67 On-chip synthesis and screening of a sialoside library yields a high affinity ligand for Siglec-7. ACS Chem Biol 2013 0.79
68 Mechanism of interaction of novel uncharged, centrally active reactivators with OP-hAChE conjugates. Chem Biol Interact 2012 0.78
69 Novel VEGFR-2 kinase inhibitors identified by the back-to-front approach. Bioorg Med Chem Lett 2013 0.78
70 A new approach to osmium-catalyzed asymmetric dihydroxylation and aminohydroxylation of olefins. Angew Chem Int Ed Engl 2002 0.78
71 Synthesis and evaluation of 1-(substituted)-3-prop-2-ynylureas as antiangiogenic agents. Bioorg Med Chem Lett 2012 0.77
72 Triazolyl tryptoline derivatives as β-secretase inhibitors. Bioorg Med Chem Lett 2010 0.77
73 Synthesis of 7-aza-5-deazapurine analogues via copper(I)-catalyzed hydroamination of alkynes and 1-iodoalkynes. J Org Chem 2010 0.77
74 Catalytic asymmetric transannulation of NH-1,2,3-triazoles with olefins. Angew Chem Int Ed Engl 2014 0.77
75 From BACE1 inhibitor to multifunctionality of tryptoline and tryptamine triazole derivatives for Alzheimer's disease. Molecules 2012 0.77
76 Interaction kinetics of oximes with native, phosphylated and aged human acetylcholinesterase. Chem Biol Interact 2010 0.76
77 Halogen exchange (Halex) reaction of 5-iodo-1,2,3-triazoles: synthesis and applications of 5-fluorotriazoles. Angew Chem Int Ed Engl 2012 0.76
78 Preparation of 1,5-Disubstituted 1,2,3-Triazoles via Ruthenium-catalyzed Azide Alkyne Cycloaddition. Organic Synth 2013 0.75
79 Ruthenium-catalyzed cycloadditions of 1-haloalkynes with nitrile oxides and organic azides: synthesis of 4-haloisoxazoles and 5-halotriazoles. Chemistry 2014 0.75
80 Synthesis and biological evaluation of furanoallocolchicinoids. J Med Chem 2014 0.75