Design, synthesis, and pharmacological evaluation of bis-2-(5-phenylacetamido-1,2,4-thiadiazol-2-yl)ethyl sulfide 3 (BPTES) analogs as glutaminase inhibitors.

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Published in J Med Chem on November 30, 2012

Authors

Krupa Shukla1, Dana V Ferraris, Ajit G Thomas, Marigo Stathis, Bridget Duvall, Greg Delahanty, Jesse Alt, Rana Rais, Camilo Rojas, Ping Gao, Yan Xiang, Chi V Dang, Barbara S Slusher, Takashi Tsukamoto

Author Affiliations

1: Department of Neurology and Brain Science Institute, Johns Hopkins University, Baltimore, Maryland 21205, United States.

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