SCH-C (SCH 351125), an orally bioavailable, small molecule antagonist of the chemokine receptor CCR5, is a potent inhibitor of HIV-1 infection in vitro and in vivo.

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Published in Proc Natl Acad Sci U S A on October 16, 2001

Authors

J M Strizki1, S Xu, N E Wagner, L Wojcik, J Liu, Y Hou, M Endres, A Palani, S Shapiro, J W Clader, W J Greenlee, J R Tagat, S McCombie, K Cox, A B Fawzi, C C Chou, C Pugliese-Sivo, L Davies, M E Moreno, D D Ho, A Trkola, C A Stoddart, J P Moore, G R Reyes, B M Baroudy

Author Affiliations

1: Schering-Plough Research Institute, Kenilworth, NJ 07033, USA.

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