Nongenomic actions of bile acids. Synthesis and preliminary characterization of 23- and 6,23-alkyl-substituted bile acid derivatives as selective modulators for the G-protein coupled receptor TGR5.

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Published in J Med Chem on August 09, 2007

Authors

Roberto Pellicciari1, Hiroyuki Sato, Antimo Gioiello, Gabriele Costantino, Antonio Macchiarulo, Bahman M Sadeghpour, Gianluca Giorgi, Kristina Schoonjans, Johan Auwerx

Author Affiliations

1: Dipartimento di Chimica e Tecnologia del Farmaco, Università di Perugia, Via del Liceo 1, 06123 Perugia, Italy. rp@unipg.it

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