Coupling of receptor conformation and ligand orientation determine graded activity.

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Published in Nat Chem Biol on October 10, 2010

Authors

John B Bruning1, Alexander A Parent, German Gil, Min Zhao, Jason Nowak, Margaret C Pace, Carolyn L Smith, Pavel V Afonine, Paul D Adams, John A Katzenellenbogen, Kendall W Nettles

Author Affiliations

1: Department of Cancer Biology, The Scripps Research Institute, Scripps Florida, Jupiter, Florida, USA.

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